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Opioid Analgesics
Indications: Managing post-operative pain, acute injury pain, cancer or palliative care pain, Non responsive pain to other mediations.
Side Effects: Constipation, sedation, nausea, respiratory depression, misuse/abuse.
Interactions: CNS Depressants will increase sedation and respiratory depression.
Fentanyl
Brand Name: Sublimate, Duragesic
Classification: Opioid Analgesic
Hydromorphone
Brand Name: Dilaudid
Classification: Opioid Analgesic
Morphine
Brand Name: MS Contin (ER), Roxanne
Classification: Opioid Analgesic
Oxycodone
Brand Name: OxyContin (ER), Roxicodone
Classification: Opioid Analgesic
Methadone
Brand Name: Dolophine
Classification: Opioid Analgesic
Codeine/Acetaminophen
Brand Name: Tylenol #3
Classification: Opioid Analgesic
Hydrocodone/Acetaminophen
Brand Name: Vicodin, Norco, Lortab
Classification: Opioid Analgesic
Tramadol
Brand Name: Ultram
Classification: Opioid Analgesic
Low-relief/extra side effects of anti-depressants
Oxycodone/Acetaminophen
Brand Name: Percocet, Endocet, Roxicet
Classification: Opioid Analgesic
Buprenorphine/Naloxone
Brand Name: Suboxone
Classification: Opioid Analgesic
Agonist/Antagonist; Lower chance of misuse
Naloxone
Brand Name: Narcan
Classification: Opioid Antagonist
Used for overdose.
Acetaminophen
Brand Name: Tylenol
Classification: Non-opioid analgesic/antipyretic
Indication: Pain&Fever
Side Effects: Hepatotoxicity (Liver)
Interactions: Alcohol, duplicate acetaminophen
Acetadote
Brand Name: Acetylcysteine
Indication: Acetaminophen overdose
Non Steroidal Anti Inflammation Drugs (NSAID)
Indications: Pain, Fever, Inflammation
Side Effects: GI Bleeding, Hypertension, Cardiovascular events, Nephrotoxicity
Interactions: Increased bleeding with anticoagulants/anti platelet and decreases hypertensive medication effectiveness.
Ibuprofen
Brand Name: Advil, Motrin
Classification: NSAID
Naproxen
Brand Name: Aleve, Naprosyn
Classification: NSAID
Diclofenac
Brand Name: Voltaren
Classification: NSAID
Indomethacin
Brand Name: Indocin
Classification: NSAID
Meloxicam
Brand Name: Mobic
Classification: NSAID
Ketorolac
Brand Name: Toradal
Classification: NSAID
Injectable 5x/Day
Celocoxib
Brand Name: Celebrex
Classification: NSAID
Lidocaine
Brand Name: Lidoderm (Patch)
Indication: Local pain relief
Side Effects: Local rash and toxicity
Triptans
Indication: Migraine
Side effects: Chest tightness, Myocardial infraction, Serotonin Syndrome, Hypertension
Interactions: Antidepressants and other drugs that increase Serotonin
Sumatriptan
Brand Name: Imitrex
Classification: Triptan
Rizatriptan
Brand Name: Maxalt
Classification: Triptan
CGRP Inhibitors
Indication: Migraine
Side Effects: Injection site reaction, Anaphylaxis
Erenumab
Brand Name: Aimovig
Classification: CGRP Inhibitor
Fremanezumab
Brand Name: Ajovy
Classification: CGRP Inhibitor
Galcanezumab
Brand Name: Emgality
Classification: CGRP inhibitor
Anticonvulsant
Indications: Seizures, Neuropathic pain, mood disorders, migraines
Side Effects: Sedation, Dizziness, Steven Johnson Syndrome
Valproic acid
Brand Name: Depakote
Classification: Anticonvulsant
Indication: Seizures, bipolar, migraine
Phenytoin
Brand Name: Dilantin
Classification: Anticonvulsant
Indication: Seizures
Lacosamide
Brand Name: Vimpat
Classification: Anticonvulsant
Indication: Seizures
Carbamazepine
Brand Name: Tegretol
Classification: Anticonvulsant
Indication: Seizures
Oxcarbazepine
Brand Name: Trileptal
Classification: Anticonvulsant
Indication: Seizures
Lamotrigine
Brand Name: Lamictal
Classification: Anticonvulsant
Indication: Seizures, Bipolar
Zonisamide
Brand Name: Zonegran
Classification: Anticonvulsant
Indication: Seizures
Levetiracetam
Brand Name: Keppra
Classification: Anticonvulsant
Indication: Seizures
Topriamate
Brand name: Topamax
Classification: Anticonvulsant
Indication: Seizures, Migrain
Pregabalin
Brand Name: Lyrica
Classification: Anticonvulsant
Indication: Neuropathic pain, Seizures
Gabapentin
Brand Name: Neurotin
Classification: Anticonvulsant
Indication: Neuropathic pain, Seizures
Anti-Parkinsons Agent
Indication: Parkinsons
Side Effects: Dyskinesias and Hallucinations
Interactions: Dopamine antagonists (antipsychotics, metoclopramide) reduce effectiveness.
Carbidopa/Levodopa
Brand Name: Sinemet
Classification: Anti-Parkinsons
Ropinirole
Brand Name: Requip
Classification: Anti-Parkinsons (DA agonist)
Also causes restless leg syndrome
Pramipexole
Brand Name: Mirapex
Classification: Anti-Parkinsons (DA agonist)
Also causes restless leg syndrome
Anti-Alzheimers drugs
Indication: Alzheimers
Side effects: Bradycardia (Oral Drugs)
Cerebral Edema/Bleeding (mABS)
Interactions:Anticholinergics oppose AChE-Is; β-blockers ↑ bradycardia
Donepezil
Brand Name: Aricept
Classification: Anti-Alzheimers (AChE-Inhibitor)
Galantamine
Brand Name: Razadyne
Classification: Anti-Alzheimers (AChE-Inhibitor)
Rivastigmine
Brand Name: Exelon
Classification: Anti-Alzheimers (AChE-Inhibitor)
Memantine
Brand Name: Namenda
Classification: Anti-Alzheimers (NMDA Antagonist)
Donepezil/Memantine
Brand Name: Namzaric
Classification: Anti-Alzheimers (AChE-Inhibitor/NMDA)
Lecanemab
Brand Name: Leqembi
Classification: Anti-Alzheimers (mAb)
Donanemab
Brand Name: Kisunla
Classification: Anti-Alzheimers (mAb)
Selective Serotonin Reuptake Inhibitor (SSRI)
Indication: Major Depressive Disorder, Anxiety Disorder
Side Effects: GI upset, headache, sexual dysfunction, Sleep disturbances, Suicidal ideation, Serotonin Syndrome
Interactions: MAOIs, Linezolid, Triptans increase risk of serotonin syndrome
Citalopram
Brand name: Celexa
Classification: SSRI
Escitalopram
Brand Name: Lexapro
Classification: SSRI
Fluoxetine
Brand Name: Prozac
Classification: SSRI
Paroxetine
Brand Name: Paxil
Classification: SSRI
Sertraline
Brand Name: Zoloft
Classification: SSRI
Serotonin Norepinephrine Reuptake Inhibitor (SNRI)
Indication: Major depressive disorder, anxiety disorder
Side Effects: GI upset, headache, sexual dysfunction, Sleep disturbances, Suicidal ideation, Serotonin Syndrome
Interactions: MAOIs, Linezolid, Triptans increase risk of serotonin syndrome
Duloxetine
Brand Name: Cymbalta
Classification: SNRI
Other Indications: Neuropathic pain
Desvenlafaxine
Brand name: Pristiq
Classification: SNRI
Venlafaxine
Brand Name: Effexor (XR)
Classification: SSRI
Tricyclic Antidepressants (TCA)
Indications: Major depressive Disorder, Anxiety Disorder
Side Effects: Anticholinergic, fatal in overdose, serotonin syndrome
Interactions: MAOIs, Linezolid, Triptans increase risk of serotonin syndrome
Amitriptyline
Brand Name: Elavil
Classification: TCA
Additional Indications: Neuropathic Pain, Migraine
Doxepin
Brand Name: Sinequan
Classification: TCA
Addictional Indications: Insomnia
Bupropion
Brand Name: Wellbutrin/Zybran
Classification: MISC.
Indications: Major Depressive Disorder, Anxiety Disorder, Smoking Cessation
Mirtazapine
Brand Name: Remeron
Classification: MISC.
Indications: Major Depressive Disorder, Anxiety Disorder
Trazodone
Brand Name: Desyrel
Classification: MISC.
Indications: Major Depressive Disorder, Anxiety Disorder, Insomnia
Antipsychotics
Indications: Schizophrenia, Bipolar, Acute Agitation
Side Effects: Extrapyramidal Symptoms, Metabolic Syndrome, QTC Prolongation
Interactions: Baseline QT Prolongation, Anti-Parkinson Drugs
Aripiprazole
Brand Name: Abilify
Classification: Antipsychotic
Quetiapine
Brand Name: Seroquel
Classification: Antipsychotic
Risperidone
Brand Name: Reisperdal
Classification: Antipsychotic
Olanzapine
Brand Name: Zyprexa
Classification: Antipsychotics
Ziprasidone
Brand Name: Geodon
Classification: Antipsychotic
Haloperidol
Brand Name: Haldol
Classification: Antipsychotic
Lithium
Indication: Mood stabilizer for bipolar
Classification: Mood Stabilizer
Brand Name: Lithobid
Side effects: Tremors, Seizures, Arrhythmias
Benzodiazepines
Schedule IV
Indication: Anxiety, Alcohol Withdrawal, Status epileptics.
Side Effects: Sedation, Respiratory depression, Abuse/Misuse, Withdrawal risk.
Interactions: Alcohol, CNS Depressants
Clonazepam
Brand Name: Klonopin
Classification: Benzodiazepine
Alprazolam
Brand Name: Xanax
Classification: Benzodiazepine
Diazepam
Brand Name: Valium
Classification: Benzodiazepine
Chlordiazepoxide
Brand Name: Librium
Classification: Benzodiazepine
Midazolam
Brand Name: Versed
Classification: Benzodiazepine
Lorazepam
Brand Name: Ativan
Classification: Benzodiazepine
Buspirone
No Regulation
Brand Name: Buspar
Classification: Non-Benzodiazepine
Indication: Anxiety
Side Effects: Serotonergic medications and Counter interactions with MAOIs
Non-Benzodiazepine Hypnotics
Schedule IV
Indication: Insomnia
Side Effects: Compex Sleep Behaviors, CNS Depression
Interactions: Alcohol, Benzodiazepines, Opioids
Eszopiclone
Brand Name: Lunesta
Classification: Non-Benzodiazepine Hypnotic
Zolpidem
Brand Name: Ambien
Classification: Non-Benzodiazepine Hypnotic
Zaleplon
Brand Name: Sonata
Classification: Non-Benzodiazepine Hypnotic
CNS Stimulants
Schedule II
Indication: ADHD
Side Effects: Insomnia, Weight loss, Cardiovascular events, hypertension, abuse/misuse
Interactions: MAOIs (Hypertensive crisis)
Amphetamine/Dextroamphetamine
Brand Name: Adderall
Classification: CNS Stimulant
Dexmethylphenidate
Brand Name: Focalin
Classification: CSN Stimulant
Methylphenidate
Brand Name: Ritalin, Concentra, Daytrana (patch)
Classification: CNS Stimulant
Lisdexamfetamine
Brand Name: Vyvanse
Classification: CNS Stimulant
Atomoxetine
Brand Name: Strattera
Classification: Non-Stimulant ADHD agent
Side Effects: Suicidal Ideation
Interaction: MAOIs for Hypertensive Crisis
General Anesthetics
Indication: cause sedation for procedures and intubation
Side Effects; Respiratory depression, Hypotension, Bradycardia
Interactions: Blood Pressure and Heart rate lowering drugs, CNS depressants
Etomidate
Brand Name: Amidate
Classification: General Anesthetics
Propofol
Brand Name: Diprivan
Classification: General Anesthetics
CI: Egg Allergy
Dexmedetomidine
Brand Name: Precedex
Classification: General Anesthetics (Light Sedation)