Targets (BUM)

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6 Terms

1
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Targets

99% Proteine

1% DNA

Sehr selten RNA oder Membran

2
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DNA als Target

Cisplastin (hemmt die Replikation)

Actinomycin D (interkalisiert in DNA, Nukleotidanalog)

3
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GPCR als Target

Morphin (µ Rezeptor)

Propanolol (ß Rezeptor / antagonist)

4
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Enzym als Target

Sildenafil (Phosphodiesterase 5)

Enalapril (Prodrug) => Enalaprilat (ACE-Hemmung)

5
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Heparin

Bindet Calcium

6
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Antacida

Neutralisieren Magen HCl

Binden H3O+