Antipsychotic receptor affinity

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10 Terms

1
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Moderate at D and also acts at 5HT1a, 5HT2a, and 5HT2c, M, and H

clozapine

2
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Interacts with 5HT2a, 5HT2c, D, M, H, and (something) 1

olanzapine

3
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Antagonists at D, 5HT, M and H

quetiapine

4
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High affinity for D receptors, some 5HT

haloperidol

5
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High affinity for 5HT2, some for D2

Antagonist at H1 and something 1 and 2

risperidone

6
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High affinity antagonist for 5HT2 and D2

ziprasidone

7
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High affinity antagonists for 5HT2 (5HT2a and 7) and D2 with some antagonist at at something 2c and 2a

partial agonist at 5HT1a

lurasidone

8
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D2 partial agonist, 5HT1 partial agonist, antagonist at 5HT2 with some monoamine reuptake inhibition

abilify

9
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Partial agonist at D2 and D3 and 5HT1a and antagonist at 5HT2a

cariprazine

10
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Partial agonist at D2 and 5HT1a and antagonist at 5HT2a

brexpiprazole