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Rifampicina
Inductor (CYP3A4, CYP2D6, UGT)
Fenitoína
Inductor
Carbamacepina
Inductor con efecto autoinductor
Efavirez
Inductor
Hierba de San Juan
Inductor
Amiodarona
Inhibidor (CYP3A4, CYP2C9, CYP2D6)
Cimetidina
Inhibidor (CYP3A4, CYP2C19, CYP1A2)
Azoles
Inhibidor
Antagonistas de calcio
Inhibidor
Macrólidos salvo azitromicina
Inhibidor (CYP3A4, CYP1A2)
Omeprazol
Inhibidor (CYP3A4, CYP2C19)
Ritonavir
Inhibidor (CYP3A4, CYP2D6)
Valproato
Inhibidor (CYP3A4)
Zumo de pomelo
Inhibidor (CYP3A4)