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Vocabulary flashcards covering adrenergic receptor drugs and their receptor actions.
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Alpha 1 Agonist
smooth muscle contraction
mydriasis (pupil dilation)
vasoconstriction in skin, mucosa and abdominal viscera
sphincter contraction of the GI tract and urinary bladder.
Alpha 2 Agonist
smooth muscle mixed effects
norepinephrine/noradrenaline inhibition
platelet activation.
Beta 1 Agonist
positive chronotropic (heart rate), dromotropic (conduction speed) and inotropic (force of cardiac contraction) effects
may increase amylase secretion
Beta 2 Agonist
smooth muscle relaxation
Epinephrine
Alpha-1 and Beta-1 agonist; broad adrenergic effects including vasoconstriction and cardiac stimulation.
Norepinephrine/Noradrenaline
Alpha-1 agonist; potent vasoconstrictor with some beta effects.
Phenylephrine
Alpha-1 agonist; vasoconstrictor often used as decongestant or to raise blood pressure.
Methoxamine
Alpha-1 agonist; increases vascular tone.
Cirazoline
Alpha-1 agonist.
Xylometazoline
Alpha-1 agonist; nasal decongestant.
Midodrine
Alpha-1 agonist; used to raise blood pressure in orthostatic hypotension.
Metaraminol
Alpha-1 agonist; increases blood pressure.
Chloroethylclonidine
Alpha-1 and Alpha-2 agonist.
Dopamine
Alpha-1 agonist & Beta-1 agonist; dose-dependent cardiovascular effects.
Acepromazine
Alpha-1 antagonist/blocker.
Alfuzosin
Alpha-1 antagonist/blocker.
Doxazosin
Alpha-1 antagonist/blocker.
Phenoxybenzamine
Alpha-1 & Alpha-2 antagonist/blocker.
Phentolamine
Alpha-1 & Alpha-2 antagonist/blocker.
Prazosin
Alpha-1 antagonist/blocker.
Tamsulosin
Alpha-1 antagonist/blocker.
Terazosin
Alpha-1 antagonist/blocker.
Trazodone
Alpha-1 & Alpha-2 antagonist/blocker.
Clomipramine
Alpha-1 antagonist/TCA.
Doxepin
Alpha-1 antagonist/TCA.
Hydroxyzine
Alpha-1 antagonist/H1 antagonist.
Agmatine
Alpha-2 agonist.
Dexmedetomidine
Alpha-2 agonist.
Medetomidine
Alpha-2 agonist.
Romifidine
Alpha-2 agonist.
Clonidine
Alpha-2 agonist.
Brimonidine
Alpha-2 agonist.
Detomidine
Alpha-2 agonist.
Lofexidine
Alpha-2 agonist.
Xylazine
Alpha-2 agonist.
Tizanidine
Alpha-2 agonist.
Guanfacine
Alpha-2 agonist.
Amitraz
Alpha-2 agonist.
Yohimbine
Alpha-2 antagonist/blocker.
Idazoxan
Alpha-2 antagonist/blocker.
Atipamezole
Alpha-2 antagonist/blocker.
Butamine
Beta-1 agonist.
Prenaline
Beta-1 agonist.
Metoprolol
Beta blocker; 1 & 2 antagonists.
Atenolol
Beta blocker; 1 & 2 antagonists.
Bisoprolol
Beta blocker; 1 & 2 antagonists.
Propranolol
Beta blocker; 1 & 2 antagonists.
Timolol
Beta blocker; 1 & 2 antagonists.
Nebivolol
Beta blocker; 1 antagonist.
Vortioxetine
Beta (Blocker) 1 antagonist.
Albuterol
Beta 2 agonist.
Bitolterol mesylate
Beta 2 agonist.
Formeterol
Beta 2 agonist.
Isoprenaline
Beta 2 agonist.
Levalbuterol
Beta 2 agonist.
Metaproterenol
Beta 2 agonist.
Salmeterol
Beta 2 agonist.
Terbutaline
Beta 2 agonist.
Ritodrine
Beta 2 agonist.
Butoxamine
Beta-2 antagonist.
Paroxetine
Beta-2 antagonist.