​6. Metabolism, Half-Life & Excretion

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6 Terms

1
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Hofmann Elimination

Cisatracurium

2
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​Renal Elimination (Muscle Relaxants)

Pancuronium (excreted unchanged in urine).

3
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​Biliary/Hepatic Excretion

Vecuronium, Rocuronium (liver/bile), Griseofulvin (biliary).

4
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​Plasma Cholinesterase Metabolism

Mivacurium and Succinylcholine.

5
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​Short Half-Life NSAIDs (<6 hrs)

Aspirin, Diclofenac, Etodolac, Ibuprofen, Indomethacin, Ketoprofen, Tolmetin, Mefenamic acid, Flufenamic acid.

6
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​Long Half-Life NSAIDs (>10 hrs)

Diflunisal, Nabumetone, Naproxen, Piroxicam, Tenoxicam, Tenidap, Phenylbutazone, Azapropazone, Sulindac.