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Fluvastatin (Lescol)
Statin
Pravastatin (Pravachol)
Statin
Lovastatin (Mevacor)
Statin
Simvastatin (Zocor)
Statin
Atorvastatin (Lipitor)
Statin
Rosuvastatin (Crestor)
Statin
Pitavastatin (Livalo)
Statin
enter cells by passive diffusion, distribute widely to tissues, and are mainly metabolized by CPY450 enzymes
Fluvastatin (Lescol)
Lovastatin (Mevacor)
Simvastatin (Zocor)
Atorvastatin (Lipitor)
Pitavastatin (Livalo)
Lipophilic statins
hepatoselective, require transporters for hepatic uptake, have limited extrahepatic distribution, and undergo minimal metabolism bf elimination
Pravastatin (Pravachol)
Rosuvastatin (Crestor)
Hydrophilic statins
zetia
Ezetimbe
Alirocumab (Praluent)
PCSK9-Inhibitor
Evolocumab (Repatha)
PCSK9-Inhibitor
Inclisiran (Leqvio)
PCSK9-Inhibitor
nicotinic acid, B-vitamin
Niacin
Cholestyramine (Questran)
Bile Acid Sequestrants
Colesevelam (Welchol)
Bile Acid Sequestrants
Colestipol (Colestid)
Bile Acid Sequestrants
Nexletol
Bempedoic acid
(Leqvio)
Inclisiran
Evkeeza
Evinacumab
Fenofibrate (Tricor, Trilipix)
Fibrates
Gemfibroozil (Lopid)
Fibrates
Lovaza (EPA + DHA)
Omega-3 Fatty Acids
Vascepa (icosapent ethyl)
Omega-3 Fatty Acids