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Nicotine
GANGLIONIC STIMULANTS: Agonist + type 1 ganglionic blocker
Vareniciline
GANGLIONIC STIMULANTS: partial agonist for (α4)3(ß2)2 receptor, full agonist for (α5)7 receptor
Tetraethylammonium (TMA)
GANGLIONIC STIMULANTS: nAchR agonist
Dimethylpheynlpiperazinium (DMPP)
GANGLIONIC STIMULANTS:nAChR agonist
Trimetaphan
Type II ganglionic blocker → non-competitive antagonist of (α3)2(ß2)3 nAChR
Hexamethonium
Type II ganglionic blocker → non-competitive antagonist of (α3)2(ß2)3 nAChR