Kaarten: CYP enzymen | Quizlet

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8 Terms

1
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CYP1A2

Substraten

warfarine, theofylline

Inhibitoren

fluvoxamine

Inductoren

carbamazepine, fenytoïne, rifampicine, sigarettenrook

2
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CYP2B6

Inductoren

carbamazepine

3
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CYP2C8

Substraten

carbamazepine

4
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CYP2C9

Substraten

acenocoumarol, fenytoïne, glibenclamide, gliclazide, glimepiride, glipizide, gliquidon, warfarine

Inhibitoren

fluconazol, miconazol

Inductoren

carbamazepine, fenytoïne, rifampicine

5
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CYP2C19

Substraten

citalopram, fenytoine, escitalopram

Inhibitoren

fluconazol, fluvoxamine

Inductoren

rifampicine

6
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CYP2D6

Substraten

codeine, flecaïnide, haloperidol, tramadol, tamoxifen

Inhibitoren

fluoxetine, paroxetine, terbinafine

Inductoren

weinig induceerbaar

7
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CYP3A4

Substraten

apixaban, atorvastatin, carbamazepine, domperidone, ethinylestradiol, oestrogenen, oestroprogestagenen, progestagenen, rivaroxaban, simvastatine, ulipristal

Inhibitoren

claritromycine, erytromycine, itraconazol,ketoconazol, pompelmoes, posaconazol, voriconazol

Inductoren

carbamazepine, rifampicine, rufinamide, sint janskruid

8
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P-gp

Substraten

apixaban, dabigatran, edoxaban, rivaroxaban (DOACs), digoxine

Inhibitoren

amiodaron

Inductoren

carbamazepine, rifampicine, sint janskruid