Adrenergic Drugs (Sympathetic Drugs)

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13 Terms

1
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Sympathetic Agonist

(α-1 Agonist)

• Phenylephrine

• Pseudoephedrine

• Xylometazoline

• Oxymetazoline

2
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Sympathetic Agonist

(α-2 Agonist)

• Clonidine

• Brimonidine

• Apraclonidine

• Methyldopa

3
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Sympathetic Agonist

(B-2 Agonist - Short Acting)

• Salbutamol

• Terbutaline

4
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Sympathetic Agonist

(B-2 Agonist - Long Acting)

• Salmeterol

• Formoterol

• Vilanterol

• Indacaterol

5
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Sympathomimetic

Mixed (a- B) Agonist

  • Epinephrine

  • Norepinephrine

  • Dopamine

6
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Sympathomimetic

Mixed B1 & B2 Agonist

• Isoproterenol

• Dobutamine

7
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Sympathetic Antagonist

a-1 Antagonist

• Doxazosin

• Terazosin

• Prazosin

• Tamsulosin

• Alfuzosin

• Silodosin

8
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Sympathetic Antagonist

a-2 Antagonist

• Mirtazapine

9
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Sympathetic Antagonist

a-1 & a-2 Mixed Antagonist

• Phentolamine (Reversible)

• Phenoxybenzamine (Irreversible)

10
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Sympathetic Antagonist

B Antagonist | Non-selective (B1 & B2)

  • Propranolol

  • Pindolol

  • Nadolol

  • Timolol

  • Levobutolol

11
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Sympathetic Antagonist

B Antagonist | Cardio Selective (B1 only)

  • Esmolol

  • Metoprolol

  • Acebutolol

  • Atenolol

  • Bisoprolol

  • Betaxolol

  • Nebivolol

12
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Sympathetic Antagonist

B Antagonist | B1,B2 & a1 Antagonist

• Labetalol

• Carvedilol

13
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Sympathetic Antagonist

B Antagonist | Partial Agonist & Antagonist (ISA)

• Acebutolol

• Pindolol

• Oxprenolol