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cocaine
Dopamine - blocks reuptake
antiosychotics
dopamine / Norepinephrine - block receptors, reducing NT availability.
Amphetamines
Dopamine / Norepinephrine - Block reuptake
Reserpine
Serotonin / Dopamine / Norepineprhine - Blocks VMAT2 vesicle
SSRIs
Serotonin - Block reuptake
Tricyclics
Serotonin - Also block reuptake
Phenelzine
Serotonin - MAO inhibitor
MDMA
Serotonin - 5-HT2 agonist
scopalamine
Acetylcholine - muscarinic receptor antagonist (motion sickness, can cross BBB)
Atropine
Acetylcholine - Muscarinic receptor Antagonist (increases heart rate)
Physostigmine
Acetylcholine - inhibits AChE, CNS
Neostigmine
Acetylcholine - inhibits AChE, treats Myasthenia gravis in PNS
AP5
glutamte - Blocks NMDA receptor, competitive agonist
Ketamine
glutamate - blocks NMDA receptor, sedative
MK-801
glutamate - blocks NMDA, noncompetitive antagonist, pore blocker
Picrotoxin
GABA - noncompetitive antagonist, convulsant
Alcohol
GABA - GABA(a) allosteric agonist
bicuculine
GABA - competitive antagonist for GABA(a)
Muscimol / ibotenic acid
GABA - GABA(a) agonist
propanolol
Norepinephrine - Beta blocker, used for ptsd.