autocoids receptor affinity drug

Prazosin, terazosin, doxazosin

Which alpha antagonist has an α₁ >>>> α₂ receptor affinity?

Phenoxybenzamine

Which alpha antagonist has an α₁ > α₂ receptor affinity?

Phentolamine

Which alpha antagonist has equal α₁ = α₂ receptor affinity?

Yohimbine, tolazoline

Which alpha antagonist has an α₂ >>> α₁ receptor affinity?

Labetalol, carvedilol

Which mixed alpha/beta antagonist has the receptor affinity β₁ = β₂ ≥ α₁ > α₂?

Metoprolol, acebutolol, alprenolol, atenolol, betaxolol, cileprolol, esmolol, nebivolol

Which beta antagonists have a β₁ >>> β₂ receptor affinity?

Propranolol, carteolol, nadolol, penbutolol, pindolol, timolol

Which beta antagonists have equal β₁ = β₂ receptor affinity?

Butoxamine

Which beta antagonist has a β₂ >>> β₁ receptor affinity?

Phenylephrine, methoxamine

Which alpha agonists have an α₁ > α₂ >>>>> β receptor affinity?

Clonidine, methylnorepinephrine

Which alpha agonists have an α₂ > α₁ >>>>> β receptor affinity?

Norepinephrine

Which mixed alpha/beta agonist has an α₁ = α₂ < β₁ >>> β₂ receptor affinity?

Epinephrine

Which mixed alpha/beta agonist has an α₁ = α₂ = β₁ = β₂ receptor affinity?

Dobutamine

Which beta agonist has a β₁ > β₂ >>>>> α receptor affinity?

Isoproterenol

Which beta agonist has a β₁ = β₂ >>>>> α receptor affinity?

Albuterol, terbutaline, metaproterenol, ritodrine

Which beta agonists have a β₂ >>> β₁ >>>>> α receptor affinity?

Dopamine

Which dopamine agonist has a D₁ = D₂ >>> β >>> α receptor affinity?

Fenoldopam

Which dopamine agonist has a D₁ >>> D₂ receptor affinity?

Phenylephrine

Which α₁ agonist is coupled to Gq, increases IP₃/DAG, and is associated with chromosome C20?

Tamsulosin

Which α₁A antagonist is associated with chromosome C8?

Clonidine

Which α₂ agonist is coupled to Gi and decreases cAMP, with the α₂ receptor effect common to all α₂ subtypes?

Yohimbine

Which α₂ antagonist is associated with the α₂ type receptor?

Oxymetazoline

Which α₂A agonist is listed in the receptor table?

Prazosin

Which α₂B antagonist is listed in the receptor table?

Prazosin

Which α₂C antagonist is listed in the receptor table?

Isoproterenol

Which β agonist is coupled to Gs and increases cAMP?

Propranolol

Which β antagonist is coupled to the β receptor system and listed with Gs?

Betaxolol

Which β₁ antagonist is associated with chromosome C10?

Butoxamine

Which β₂ antagonist is associated with chromosome C5?

Mirabegron

Which β₃ agonist is associated with chromosome C8?

Fenoldopam

Which D₁ agonist is coupled to Gs and increases cAMP, with the gene on chromosome C5?

Bromocriptine

Which D₂ agonist is coupled to Gi and decreases cAMP, with the gene on chromosome C11?

Clozapine

Which D₄ antagonist is coupled to Gi and decreases cAMP, with the gene on chromosome C11?

D₃

Which dopamine receptor is coupled to Gi and decreases cAMP, with the gene on chromosome C3?

D₅

Which dopamine receptor is coupled to Gs and increases cAMP, with the gene on chromosome C