Cytochrome P450, CYP3A4 Substrates, Inhibitors, and Inducers

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P450

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77 Terms

1
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Alfentanil

Substrate

2
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Aliskiren

Substrate

3
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Alphazolam

Substrate

4
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amiodarone

Substrate

Inhibitor

5
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Amlodipine

Substrate

Inhibitor

6
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Apixaban

Substrate

7
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Aripiprazole

Substrate

8
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Atorvastatin

Substrate

9
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Brexpiprazole

Substrate

10
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Budesonide

Substrate

11
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Buprenorphine

Substrate

12
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Buspirone

Substrate

13
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Carbamazepine

Substrate

Inducer

14
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Colchicine

Substrate

15
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Dexamethasone

Substrate

Inducer

<p>Substrate</p><p>Inducer</p>
16
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Diazepam

Substrate

17
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Diltiazem

Substrate

Inhibitor

18
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Domperidone

Substrate

19
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Dronedarone

Substrate

Inhibitor

20
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Eplerenone

Substrate

21
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Esomeprazole

Substrate

22
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Estrogens

Substrate

23
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Ethinyl Estradiol

Substrate

Inhibitor

24
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Etonogestrel

Substrate

25
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Felodipine

Substrate

26
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Fentanyl

Substrate

27
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Fluticasone

Substrate

28
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Haloperidol

Substrate

29
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Hydrocodone

Substrate

30
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Itraconazole

Substrate

31
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Ketoconazole

Substrate

32
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Levonorgestrel

Substrate

33
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Linagliptin

Substrate

34
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Lovastatin

Substrate

35
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Lurasidone

Substrate

36
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Methadone

Substrate

37
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Methylprednisolone

Substrate

38
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Nifedipine

Substrate

39
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Omeprazole

SubstrateO

40
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Oral Contraceptives

Substrate

41
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Oxycodone

Substrate

42
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Quetiapine

Substrate

43
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Risperidone

Substrate

44
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Salmeterol

Substrate

45
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Saxagliptin

Substrate

46
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Sildenal

Substrate

47
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Simvastatin

Substrate

48
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Tramadol

Substrate

49
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Trazodone

Substrate

50
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Verapamil

Substrate

51
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Voriconazole

Substrate

52
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(R) Warfarin

Substrate

53
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Zolpidem

Substrate

54
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Cimetidine

Inhibitor

55
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Ciprofloxacin

Inhibitor

56
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Clarithromycin

Inhibitor

57
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Cobicistat

Inhibitor

58
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Erythromycin

Inhibitor

59
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Fluconazole

Inhibitor

60
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Fluoxetine

Inhibitor

61
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Fluvoxamine

Inhibitor

62
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Grapefruit

Inhibitor

63
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Lansoprazole

Inhibitor

64
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Nefazodone

Inhibitor

65
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Nicardipine

Inhibitor

66
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Posaconazole

Inhibitor

67
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Synercid

Inhibitor

68
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Voriconazole

Inhibitor

69
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Modafinil

Inducer

70
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Nafcillin

Inducer

71
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Oxcarbazepine

Inducer

72
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Phenobarbital

Inducer

73
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Phenyotin

Inducer

74
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Rifampin

Inducer

75
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Rifapentine

Inducer

76
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St. John’s Wort

Inducer

77
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Topiramate

Inducer

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