Smoking Cessation

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10 Terms

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Varenicline MOA

partial a/B2 nicotinic agonist that stimulates dopamine to a much smaller degree than nicotine

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Varenicline indications

smoking cessation

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Varenicline dosage forms

oral

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Varenicline administration

after eating and with a full glass of water

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Varenicline major side effects

CV events, nausea, vomiting, disordered sleep, insomnia, irritability, neuropsychiatric events, seizures

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Varenicline safety monitoring parameters

mental status changes

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Varenicline efficacy monitoring parameters

abstinence from tobacco

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Varenicline major interactions

alcohol, nicotine

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Varenicline can cause

CNS depression (decreased mental alertness)

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caution Varenicline use in pts with

renal impairment