Cytochrome interactions (Alaa Nasr)

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21 Terms

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Inducers

Cause therapeutic failure of other drugs

2
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Inducers

Anti-epileptic except VPA

Rifampin

St. John’s Wart

Tobacco/Nicotine (smoking)

Barbiturates

3
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Inhibitors

Causes toxicity of other drugs

4
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Inhibitor

Valproic acid

Ciprofloxacin, Moxifloxacin

Erythromycin, Clarithromycin

Azoles

Verapamil, Diltiazem

Cimetidine

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Cimetidine

1A2, 2C9, 2D6 inhibitor

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Paroxetine

2D6 inhibitor

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Verapamil

Amiodarone

Diltiazem

Clarithromycin

Grapefruit juice

Erythromycin

3A4 inhibitor

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Amiodarone

3A4, 2C9, 2D6 inhibitor

9
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Smoking

Tobacco

1A2 inducer

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Rifampicin

3A4, 2C9 inducer

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Codeine

2D6 substrate

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Rivaroxaban

Apixaban

Verapamil

Colchicine

Metabolised by 3A4

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Digoxin

3A4 substrate

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Phenytoin

Irbesartan

Metabolised by 2C9

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Clopidogrel

Prodrug activated by 2C19

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Ibuprofen

Celecoxib

Losartan

Phenytoin

2C9 substrate

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90% 1A2, 10% 3A4

Lidocaine metabolism

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Bupropion

2B6 substrate, 2D6 inhibitor

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NSAID (especially ibuprofen)

Measures 2C9

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Erythromycin

Measures 3A4

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Dextrometorphan

Measures 2D6