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inhibitory or excitatory: ACETYLCHOLINE
excitatory
inhibitory or excitatory: DOPAMINE
mixed (inhibitory/excitatory)
inhibitory or excitatory: NOREPINEPHRINE
excitatory
inhibitory or excitatory: SEROTONIN
inhibitory
inhibitory or excitatory: GABA
inhibitory
inhibitory or excitatory: GLYCINE
inhibitory
inhibitory or excitatory: GLUTAMATE
excitatory
inhibitory or excitatory: ASPARTATE
excitatory
inhibitory or excitatory: SUBSTANCE P
excitatory
inhibitory or excitatory: ENKEPHALINS
inhibitory
indications baclofen
MS, CP, SCI
tizanidine indications
sci spasticity
clonidine indications
hypertension, adhd
clonazepam indications
myoclonic, absence seizures, panic disorder
dantrolenea indications
tbi, cp, stroke, malignant hyperthermia
diazepam indications
muscle spasm, spasticity, anxiety, status epelipticus
botulinum toxin indications
chronic migraine, focal spasticity, cosmetics
benzodiapines (anxiolytics) moa
increases frequency of Cl channel opening, induces hyperpolarization
non benzodiazepines (anxiolytics) moa
buspirones: partial agonist 5HT1a, Z drugs: selectively bind to a1 subunit of GABA A receptor
barbiturates (anxiolytics)
binds to GABA A, prolongs Cl channel opening
MOA baclofen
GABA B receptor agonist
inhibits mono/polysynaptic reflexes
blocks release of excitatory neurotransmitter
MOA tizanidine
a2 adrenergic receptor agonist
stimulated in brainstem
blocks release of excitatory neurotransmitter
clonidine MOA
a2 adrenergic receptor agonist
acts centrally
reduces CNS output/flow
clonazepam MOA
activates GABA receptor
increases chloride ions in post synaptic cell
reduces action potentials = reduces mono/polysynaptic reflexes
dantrolenea MOA
inhibits Ca2+ release from SR
blocks ryanodine receptors
inhibits muscle contraction
botulinum toxin
prevents ACh release from presynaptic membrane
muscle contractions decrease/calmer
cleavage of SNARE protein complex (SNAP 25)
diazepam MOA
enhances GABA A for (inhibitory effects of) GABA
increased Cl- flow