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Orlistat
MOA: Pancreatic lipase inhibitor
Side Effects: Steatorrhea, oily spotting, fecal urgency, fecal incontinence
Lorcaserin
MOA: 5-HT2 serotonin agonist: reduces food intake
Side Effects: Headache, nausea, dizziness, dry mouth, constipation
Phentermine–topiramate ER
MOA: Sympathomimetic anticonvulsant: reduces food intake
Side Effects: Insomnia, dry mouth, constipation, paresthesias, dizziness, dysgeusia
Naltrexone SR-buporpion
MOA: Opioid receptor antagonist: reduces food intake
Side Effects: Nausea, vomiting, headache, constipation, dizziness
Liraglutide (Saxenda™)
MOA: GLP-1 receptor agonist: reduces food intake
Side Effects: Nausea, vomiting, diarrhea, constipation, headache, dyspepsia, fatigue, dizziness, abdominal pain
Semaglutide (Wegovy™)
MOA: GLP-1
Side Effects: Nausea, vomiting, diarrhea, constipation, headache, dyspepsia, fatigue, dizziness, abdominal pain
Setmelanotide (IMCIVREE™)
MOA: Only approved for genetic conditions (POMC deficiency; PCSK1 deficiency); leptin receptor deficiency; Bardet-Biedl syndrome)
Tirzepatide (Zepbound™)
MOA: Mimics GIP, GLP-1
Side Effects: Nausea, vomiting, diarrhea, constipation, headache, dyspepsia, fatigue, dizziness, abdominal pain