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Atorvastatin
Brands = Lipitor
Drug Class = Statin
Typical Uses = ↓ CV Events
Lovastatin
Brands = Mevacor, Altoprev
Drug Class = Statin
Typical Uses = ↓ CV Events
Pravastatin
Brands = Pravachol
Drug Class = Statin
Typical Uses = ↓ CV Events
Rosuvastatin
Brands = Crestor
Drug Class = Statin
Typical Uses = ↓ CV Events
Simvastatin
Brands = Zocor
Drug Class = Statin
Typical Uses = ↓ CV Events
Ezetimibe/Simvastatin
Brands = Vytorin
Drug Class = Combo (Chol-abs inhib + statin)
Typical Uses = ↓ CV Events
Ezetimibe
Brands = Zetia
Drug Class = Cholesterol-absorption inhibitor
Typical Uses = ↓LDL
Fenofibrate
Brands = Tricor
Drug Class = Fibrate
Typical Uses = ↓TG, ↑HDL
Gemfibrozil
Brands = Lopid
Drug Class = Fibrate
Typical Uses = ↓TG, ↑HDL
Omega-3-acid ethyl esters
Brands = Lovaza
Drug Class = Omega-3 FA (Fish Oil)
Typical Uses = ↓TG
Niacin (ER)
Brands = Niaspan
Drug Class = Vitamin B3
Typical Uses = ↑HDL, ↓TG/LDL
Alirocumab
Brands = Praluent
Drug Class = PCSK9 inhibitor
Typical Uses = ↓LDL (inject)
Evolocumab
Brands = Repatha
Drug Class = PCSK9 inhibitor
Typical Uses = ↓LDL (inject)
Mechanism / Therapeutic Rationale
• Statins: dramatic LDL-C drop. ✓ mortality benefit
• Ezetimibe: ↓cholesterol absorption; add-on to statins.
• Fibrates: ↓TG, modest ↑HDL.
• Niacin: ↑HDL, ↓TG.
• Omega-3 FA: ↓hepatic TG.
• PCSK9i: profound LDL-C ↓
Hallmark Common SEs
• Statins: GI upset, myalgias
• Fibrates: dyspepsia
• Niacin: flushing
• Omega-3: fishy taste, GI
• PCSK9i: injection-site erythema
Serious / Black-Box Risks
Statins/Fibrates/Niacin/Ezetimibe (+statin): myopathy → rhabdomyolysis
Hepatotoxicity (statins, niacin, fibrates) – monitor LFTs
PCSK9i: hypersensitivity / anaphylaxis (rare)
High-Yield Interactions & Contra-Indications
• CYP3A4 inhibitors (azoles, macrolides, grapefruit juice) ↑ ator-/sim-/lova-statin levels → myopathy.
• Fibrates markedly ↑ statin myopathy risk – avoid combo.
• Absolute CI: active liver disease, pregnancy (statins); seafood allergy (omega-3).