Hu CNS Stimulants

Drug Name and Class

Xanthine

Methylxanthine Alkaloid

Drug Name and Class

Caffeine

Methylxanthine Alkaloid

Drug Name and Class

Theophylline

Methylxanthine Alkaloid

Drug Name and Class

Theobromine

Methylxanthine Alkaloid

Drug Name and Class

Pamabrom, Diurex Max

Methylxanthine Derivative

Drug Name and Class

Aminophylline, Phyllocontin, Truphylline

Methylxanthine Derivative

Drug Name and Class

Oxtriphylline, Choledyl SA (ER tablets)

Methylxanthine Derivative

Drug Name and Class

Dyphylline, Dilor, Lufyllin

Methylxanthine Derivative

Drug Name and Class

Doxapram Hydrochloride, Dopram

Miscellaneous stimulant

Drug Name and Class

Modafinil, Provigil

Miscellaneous stimulant

Drug Name and Class

Armodafinil, Nuvigil

Miscellaneous stimulant

Drug Name and Class

Pitolisant hydrochloride, Wakix

Miscellaneous stimulant

Drug Name and Class

Solriamfetol, Sunosi

Miscellaneous stimulant

Drug Name and Class

Sodium Oxybate, Xyrem

Miscellaneous stimulant

Drug Name and Class

Dextroamphetamine Sulfate, Dexedrine

β-Phenethylamines Used Mainly as Stimulants

Drug Name and Class

Methamphetamine Hydrochloride, Desoxyn

β-Phenethylamines Used Mainly as Stimulants

Drug Name and Class

Phentermine Hydrochloride, Phentrol® Phentermine Ion-Exchange Resin, Ionamin

β-Phenethylamines Used Mainly as Anorexiants

Drug Name and Class

Benzphetamine HCl, Didrex

β-Phenethylamines Used Mainly as Anorexiants

Drug Name and Class

Diethylpropion Hydrochloride, Tenuate

β-Phenethylamines Used Mainly as Anorexiants

Drug Name and Class

Phendimetrazine Tartrate, Plegine

β-Phenethylamines Used Mainly as Anorexiants

Drug Name and Class

Orlistat, Xenical, Alli

β-Phenethylamines Used Mainly as Anorexiants

Drug Name and Class

Methylphenidate Hydrochloride, Ritalin

Attention Deficit Hyperactivity Disorder (ADHD)

Drug Name and Class

Dexmethylphenidate Hydrochloride, Focalin

Attention Deficit Hyperactivity Disorder (ADHD)

Drug Name and Class

Serdexmethylphenidate, as part of Azstarys

Attention Deficit Hyperactivity Disorder (ADHD)

Drug Name and Class

Lisdexamfetamine Dimesylate, Vyvanse

Attention Deficit Hyperactivity Disorder (ADHD)

Drug Name and Class

Atomoxetine HCl, Strattera

Attention Deficit Hyperactivity Disorder (ADHD)

Drug Name and Class

Viloxazine Hydrochloride, Qelbree

Attention Deficit Hyperactivity Disorder (ADHD)

Drug Name and Class

Phenelzine Sulfate, Nardil

Monoamine Oxidase Inhibitors (MAOI)

Drug Name and Class

Isocarboxazid, Marplan

Monoamine Oxidase Inhibitors (MAOI)

Drug Name and Class

Tranylcypromine Sulfate, Parnate

Monoamine Oxidase Inhibitors (MAOI)

Drug Name and Class

Selegiline, Emsam® Zelapar

Monoamine Oxidase Inhibitors (MAOI)

Drug Name and Class

Rasagiline, Azilect

Monoamine Oxidase Inhibitors (MAOI)

Drug Name and Class

Imipramine, Tofranil

Azepine Tricyclic Antidepressants (TCAs)

Drug Name and Class

Desipramine, Norpramin

Azepine Tricyclic Antidepressants (TCAs)

Drug Name and Class

Trimipramine Maleate, Surmontil

Azepine Tricyclic Antidepressants (TCAs)

Drug Name and Class

Clomipramine Hydrochloride, Anafranil

Azepine Tricyclic Antidepressants (TCAs)

Drug Name and Class

Amitriptyline Hydrochloride, Elavil

Cycloheptane Tricyclic Antidepressants (TCAs)

Drug Name and Class

Nortriptyline Hydrochloride, Aventyl®, Pamelor

Cycloheptane Tricyclic Antidepressants (TCAs)

Drug Name and Class

Protriptyline Hydrochloride, Vivactil

Cycloheptane Tricyclic Antidepressants (TCAs)

Drug Name and Class

Doxepin Hydrochloride, Sinequan®, Adapin

Other Heterocycles, TCAs

Drug Name and Class

Amoxapine, Asendin

Other Heterocycles, TCAs

Drug Name and Class

Maprotiline Hydrochloride, Ludiomil

Tetracyclic TCAs

Drug Name and Class

Mirtazapine, Remeron

Tetracyclic TCAs

Drug Name and Class

Fluoxetine, Prozac

Selective Serotonin Reuptake Inhibitors (SSRIs)

Drug Name and Class

Paroxetine, Paxil

Selective Serotonin Reuptake Inhibitors (SSRIs)

Drug Name and Class

Sertraline Hydrochloride, Zoloft

Selective Serotonin Reuptake Inhibitors (SSRIs)

Drug Name and Class

Fluvoxamine Maleate, Luvox

Selective Serotonin Reuptake Inhibitors (SSRIs)

Drug Name and Class

Citalopram Hydrobromide, Celexa

Selective Serotonin Reuptake Inhibitors (SSRIs)

Drug Name and Class

Escitalopram Oxalate, Lexapro

Selective Serotonin Reuptake Inhibitors (SSRIs)

Drug Name and Class

Duloxetine Hydrochloride, Cymbalta

Atyptical Antidepressants: Serotonin and Norepinephrine Reuptake Inhibitors (SNRI)

Drug Name and Class

Venlafaxine, Effexor

Atyptical Antidepressants: Serotonin and Norepinephrine Reuptake Inhibitors (SNRI)

Drug Name and Class

Desvenlafaxine, Pristiq

Atyptical Antidepressants: Serotonin and Norepinephrine Reuptake Inhibitors (SNRI)

Drug Name and Class

Levomilnacipran, Fetzima

Atyptical Antidepressants: Serotonin and Norepinephrine Reuptake Inhibitors (SNRI)

Drug Name and Class

Trazodone, Desyrel

Serotonin Antagonist at 5H2A receptor and reuptake inhibitor (SARI)

Drug Name and Class

Nefazodone, Serzone

SARI and 5-HT1A agonist (Also decreases NE reuptake)

Drug Name and Class

Vilazodone, Viibryd

SSRI + 5-HT1A partial agonist

Drug Name and Class

Vortioxetine, Brintellix

Miscellaneous Antidepressant (5-HT1A agonist + 5-HT3 antagonist)

Drug Name and Class

Bupropion Hydrochloride, Wellbutrin

Miscellaneous Antidepressant (NDRI)

Drug Name and Class

Sumatriptan, Imitrex

Serotonin 5-HT1B / 1D / 1F Receptor Agonist

Drug Name and Class

Rizatriptan, Maxalt

Serotonin 5-HT1 Receptor Agonists

Drug Name and Class

Zolmitriptan, Zomig

Serotonin 5-HT1 Receptor Agonists

Drug Name and Class

Almotriptan, Axert

Serotonin 5-HT1 Receptor Agonists

Drug Name and Class

Eletriptan, Relpax

Serotonin 5-HT1 Receptor Agonists

Drug Name and Class

Naratriptan, Amerge

Serotonin 5-HT1 Receptor Agonists

Drug Name and Class

Frovatriptan, Frova

Serotonin 5-HT1 Receptor Agonists (5-HT1F selective)

Drug Name and Class

Lasmiditan, Reyvow

Serotonin 5-HT1 Receptor Agonist

Drug Name and Class

Ubrogepant, Ubrelvy

Non-peptide small molecule CGRP receptor antagonists

Drug Name and Class

Atogepant, Qulipta

Non-peptide small molecule CGRP receptor antagonists

Drug Name and Class

Rimegepant, Nurtec ODT

Non-peptide small molecule CGRP receptor antagonists

Drug Name and Class

Zavegepant hydrochloride, Zavzpret

Non-peptide small molecule CGRP receptor antagonists

Drug Name and Class

Ondansetron Hydrochloride, Zofran

5-HT3 Receptor Antagonists as Antiemetics

Drug Name and Class

Palonosetron Hydrochloride, Aloxi

5-HT3 Receptor Antagonists as Antiemetics

Drug Name and Class

Granisetron Hydrochloride, Kytril

5-HT3 Receptor Antagonists as Antiemetics

Drug Name and Class

Alosetron Hydrochloride, Lotronex

5-HT3 Receptor Antagonists for IBS in women

Drug Name and Class

Aprepitant, Emend

Substant P Antagonist

Drug Name and Class

Rolapitant, Varubi

Substant P Antagonist

Drug Name and Class

Netupitant/palonosetron

Selective NKIR antagonist

Drug Name and Class

Fosnetupitant/palonosetron (Akynzeo®)

NKIR selective antagonist

Drug Name and Class

Dronabinol, Marinol®, Syndros

Cannabinoid

Drug Name and Class

Metoclopramide, Reglan

D2 antagonist, mixed 5-HT3 antagonist and 5-HT4 Agonist