3: Drug Classes

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Last updated 2:06 AM on 7/3/26
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327 Terms

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Zidovudine (AZT)
NRTI (Nucleoside Reverse Transcriptase Inhibitor)
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Lamivudine
NRTI
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Emtricitabine
NRTI
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Abacavir
NRTI
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Tenofovir (TDF, TAF)
NRTI / Nucleotide Reverse Transcriptase Inhibitor
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Efavirenz
NNRTI (Non-Nucleoside Reverse Transcriptase Inhibitor)
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Nevirapine
NNRTI
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Rilpivirine
NNRTI
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Doravirine
NNRTI
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Darunavir
Protease Inhibitor (PI)
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Atazanavir
Protease Inhibitor
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Lopinavir
Protease Inhibitor (often co-formulated with ritonavir)
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Ritonavir
Protease Inhibitor / pharmacokinetic booster
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Dolutegravir
Integrase Strand Transfer Inhibitor (INSTI)
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Bictegravir
INSTI
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Raltegravir
INSTI
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Elvitegravir
INSTI
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Phenobarbital
Barbiturate AED
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Phenytoin (Dilantin)
AED (sodium-channel modulator)
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Carbamazepine (Tegretol)
AED (sodium-channel modulator)
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Valproate / Valproic Acid
BROADEST-spectrum AED
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Gabapentin
AED / GABA analogue
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Ethosuximide
AED
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Clonazepam (Rivotril)
Benzodiazepine AED
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Vigabatrin
Newer AED, used in combo
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Tiagabine
Newer AED, used in combo
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Lamotrigine (Lamictal)
Newer AED, used in combo
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Topiramate
Newer AED, used in combo
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Diazepam (Valium)
Long-acting benzodiazepine
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Lorazepam (Ativan)
Intermediate-half-life benzodiazepine
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Chlorpromazine
Typical (1st-gen) antipsychotic — prototype
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Haloperidol (Haldol)
Typical antipsychotic (high- potency)
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Clozapine
Atypical antipsychotic
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Olanzapine
Atypical antipsychotic
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Risperidone (Risperdal)
Atypical antipsychotic — entry-level psychosis
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Sertindole (Serlect)
Atypical antipsychotic
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Quetiapine (Seroquel)
Atypical antipsychotic
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Ziprasidone (Geodon)
Atypical antipsychotic
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Aripiprazole (Abilify)
Atypical antipsychotic (D2 partial agonist)
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Procyclidine
Anticholinergic
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Benztropine
Anticholinergic
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Disulfiram (Antabuse)
Alcohol-sensitising agent
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Naltrexone (ReVia)
Opioid receptor antagonist (mu, kappa, delta)
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Acamprosate (Campral)
Anti-craving agent
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Ondansetron (Zofran)
5-HT₃ receptor antagonist
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Methadone
Full μ-opioid agonist
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Buprenorphine
Partial μ-opioid agonist
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Modafinil
Wakefulness-promoting agent
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Amitriptyline (Elavil)
TCA (Tricyclic Antidepressant)
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Imipramine (Tofranil)
TCA
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Trimipramine (Surmontil)
TCA
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Nortriptyline (Aventyle)
TCA
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Protriptyline (Vivactil)
TCA
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Desipramine (Pertofrane)
TCA
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Fluoxetine (Prozac)
SSRI — prototype
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Sertraline (Zolof)t
SSRI
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Paroxetine (Paxil)
SSRI
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Fluvoxamine (Luvox)
SSRI
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Citalopram (Celexa)
SSRI
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Phenelzine (Nardil)
MAOI
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Tranylcypromine (Parnate)
MAOI
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Selegiline (Eldepryl)
Selective MAO-B inhibitor
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Venlafaxine (Effexor)
SNRI
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Bupropion (Wellbutrin / Zyban)
NDRI
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Trazodone
SARI (Serotonin Antagonist / Reuptake Inhibitor)
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St. John's Wort (Hypericum perforatum)
Herbal antidepressant
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Lithium
Mood stabiliser
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Levodopa / Carbidopa
Dopamine precursor + peripheral decarboxylase inhibitor
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Amantadine
Dopamine releaser / NMDA antagonist
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Bromocriptine
Dopamine D2 agonist (ergot)
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Pergolide
D2 agonist
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Pramipexole ("Primipexole")
D2 agonist
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Ropinirole ("Ropinorole")
D2 agonist
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Rasagiline
Selective MAO-B inhibitor
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Biperiden
Anticholinergic
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Orphenadrine
Anticholinergic
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Alprazolam (Xanax)
Benzodiazepine (short half- life)
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Bromazepam (Lectopam)
Benzodiazepine
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Oxazepam (Serax)
Benzodiazepine (no Phase I metabolism)
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Chlordiazepoxide (Librium)
Benzodiazepine
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Clorazepate (Tranxene)
Benzodiazepine (PRODRUG)
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Nitrazepam (Mogadon)
Benzodiazepine
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Temazepam (Restoril)
Benzodiazepine
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Triazolam (Halcion)
Benzodiazepine (very short half-life)
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Flurazepam (Dalmane)
Benzodiazepine
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Midazolam (Versed)
Benzodiazepine (short, very lipophilic)
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Remimazolam
Ultra-short-acting benzodiazepine
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Flumazenil
Benzodiazepine antagonist
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Baclofen
GABA-B receptor agonist
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Tizanidine
α2-adrenergic agonist (similar to clonidine)
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Pregabalin
GABA analogue (Ca-channel binder)
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Procainamide
Class Ia (Na⁺-channel blocker)
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Quinidine
Class Ia
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Disopyramide
Class Ia
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Lidocaine
Class Ib (Na-channel blocker) + amide local anesthetic
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Mexiletine
Class Ib
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Flecainide
Class Ic
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Propranolol
Class II β-blocker (non- selective)
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Esmolol
Class II β-blocker (cardioselective β1, ultra- short)