Muscarinic Agonists and Antagonists

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18 Terms

1
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Acetylcholine

Agonist

Short duration

<p>Agonist</p><p>Short duration</p>
2
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Bethanechol

Agonist

Long duration

<p>Agonist</p><p>Long duration</p>
3
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Muscarine

Agonist

<p>Agonist</p>
4
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Cevimeline

Agonist

M1/M3 selective

Crosses membranes while uncharged, then binds agonist as charged

CYP 2D6

<p>Agonist</p><p>M1/M3 selective</p><p>Crosses membranes while uncharged, then binds agonist as charged</p><p>CYP 2D6</p>
5
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Atropine - 1

Antagonist

<p>Antagonist</p>
6
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Atropine - 2

Antagonist

<p>Antagonist</p>
7
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Hyoscyamine

Antagonist

Enantiomer of atropine

<p>Antagonist</p><p>Enantiomer of atropine</p>
8
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Tropicamide

Antagonist

<p>Antagonist</p>
9
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Scopolamine

Antagonist

Crosses BBB

<p>Antagonist</p><p>Crosses BBB</p>
10
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Benztropine

Antagonist

Crosses BBB

<p>Antagonist</p><p>Crosses BBB</p>
11
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Glycopyrronium bromide

Antagonist

<p>Antagonist</p>
12
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Solifenacin

Antagonist

69% unchanged in the urine

CYP 3A4

<p>Antagonist</p><p>69% unchanged in the urine</p><p>CYP 3A4</p>
13
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Oxybutynin

Antagonist

Very non-polar, can penetrate skin

<p>Antagonist</p><p>Very non-polar, can penetrate skin</p>
14
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Dicyclomine

Antagonist

<p>Antagonist</p>
15
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Tiotropium bromide

Antagonist

M1 selective

Long acting

Protonated amine means it stays in the lungs

<p>Antagonist</p><p>M1 selective</p><p>Long acting</p><p>Protonated amine means it stays in the lungs</p>
16
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Ipratropium bromide

Antagonist

M1 selective

Protonated amine means it stays in the lungs

<p>Antagonist</p><p>M1 selective</p><p>Protonated amine means it stays in the lungs</p>
17
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Trospium

Antagonist

<p>Antagonist</p>
18
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Xanomeline

Agonist

Crosses BBB

<p>Agonist</p><p>Crosses BBB</p>