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D2 Antagonists / Haloperidol
Most effective for tics & decrease DA overactivity
SSRIs / Fluoxetine/Sertraline/Clomipramine
treat OCD symptoms
Botulinum Toxin (TS)
focal/disabling tics
Botulinum Toxin (dystonia)
Act at NMJ
Inhibits ACh exocytosis by cleaving SNARE proteins (SNAP-25, VAMP, syntaxin) → chemical denervation
Treatment of choice for focal dystonia
Resistance due to antibodyformation
Baclofen
act at SC
GABA-B agonist → presynaptic inhibition
Intrathecal in severe dystonia
Anticholinergics
Act at CNS & NMJ
Muscarinic receptor antagonists
First-line adults (Children: L-DOPA first)
Lose efficacy = circuitadaptation
Benzodiazepines
Act at CNS
GABA-A agonists
Less effective; sedation