FFM2 Mini 2

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Last updated 8:31 PM on 8/7/26
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68 Terms

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Catecholamine (direct-acting) agonists
Adrenergic agonists
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Epinephrine
Agonist at α₁, α₂, β₁, β₂ receptors
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Norepinephrine
Agonist at α₁, α₂, β₁ receptors
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Isoproterenol
Agonist at β₁, β₂ receptors
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Dobutamine
Agonist at β₁ receptors
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Dopamine
Agonist at D₁ receptors (β₁ & α₁ at high doses)
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Non-catecholamine agonists
Selective adrenergic agonists
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Phenylephrine, Oxymetazoline, Methoxamine
α₁ agonists
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Albuterol, Pirbuterol, Terbutaline, Salmeterol, Formoterol
β₂ agonists
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Metaproterenol
β₂ > β₁ agonist
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Clonidine, Apraclonidine
α₂ agonists
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Ephedrine, Pseudoephedrine
Mixed α & β agonists
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α-Adrenergic Antagonists (α-Blockers)
Phentolamine (competitive/reversible), Phenoxybenzamine (irreversible), Prazosin, Terazosin, Doxazosin, Tamsulosin (α₁A-selective), Silodosin, Yohimbine, Mirtazapine
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Nonselective α-blockers
Phentolamine (competitive/reversible), Phenoxybenzamine (irreversible)
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α₁-Selective blockers
Prazosin, Terazosin, Doxazosin, Tamsulosin (α₁A-selective), Silodosin
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α₂-Selective blockers
Yohimbine, Mirtazapine
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β-Adrenergic Antagonists (β-Blockers)
Propranolol, Timolol, Sotalol, Nadolol, Atenolol, Metoprolol, Esmolol, Acebutolol, Pindolol, Labetalol, Carvedilol
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Non-selective β-blockers (no ISA)
Propranolol, Timolol, Sotalol, Nadolol
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β₁-selective blockers
Atenolol, Metoprolol, Esmolol, Acebutolol
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Beta antagonist with intrinsic sympathomimetic activity (ISA)

Pindolol, Acebutolol

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Combined α/β-blockers
Labetalol, Carvedilol
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Direct-acting cholinergic drugs – Muscarinic agonists
Direct muscarinic receptor agonists
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Pilocarpine
Muscarinic agonist
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Muscarine
Muscarinic agonist
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Bethanechol
Muscarinic agonist
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Carbachol
Muscarinic and nicotinic agonist
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Acetylcholine
Muscarinic and nicotinic agonist
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Direct-acting cholinergic drugs – Nicotinic agonists
Direct nicotinic receptor agonists
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Nicotine
Nicotinic agonist
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Indirect-acting cholinergic drugs – Cholinesterase inhibitors
Acetylcholinesterase inhibitors (indirect cholinergic agonists)
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Edrophonium
Reversible acetylcholinesterase inhibitor
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Physostigmine
Reversible acetylcholinesterase inhibitor
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Pyridostigmine
Reversible acetylcholinesterase inhibitor
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Neostigmine
Reversible acetylcholinesterase inhibitor
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Donepezil
Reversible acetylcholinesterase inhibitor
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Parathion
Irreversible acetylcholinesterase inhibitor (organophosphate)
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Malathion
Irreversible acetylcholinesterase inhibitor (organophosphate)
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Pralidoxime (2-PAM)
Cholinesterase reactivator (reactivates acetylcholinesterase after organophosphate poisoning)
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Natural alkaloids
Antimuscarinic agents
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Atropine
Antimuscarinic (tertiary amine)
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Scopolamine
Antimuscarinic (tertiary amine)
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Synthetic tertiary amines
Antimuscarinic agents
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Homatropine
Antimuscarinic (tertiary amine)
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Oxybutynin
Antimuscarinic (tertiary amine)
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Cyclopentolate
Antimuscarinic (tertiary amine)
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Tropicamide
Antimuscarinic (tertiary amine)
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Dicyclomine
Antimuscarinic (tertiary amine)
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Pirenzepine
Antimuscarinic (tertiary amine)
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Tolterodine
Antimuscarinic (tertiary amine)
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Synthetic quaternary ammonium compounds
Antimuscarinic agents
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Glycopyrrolate
Antimuscarinic (quaternary ammonium)
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Ipratropium
Antimuscarinic (quaternary ammonium)
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Tiotropium
Antimuscarinic (quaternary ammonium)
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Antiparkinsonian agents
Antimuscarinic agents
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Trihexyphenidyl
Antimuscarinic (tertiary amine)
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Procyclidine
Antimuscarinic (tertiary amine)
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Benztropine
Antimuscarinic (tertiary amine)
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Non-depolarizing ganglionic blockers
Ganglionic nicotinic receptor antagonists
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Hexamethonium
Non-depolarizing ganglionic blocker
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Trimethaphan
Non-depolarizing ganglionic blocker
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Mecamylamine
Non-depolarizing ganglionic blocker
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Depolarizing NMJ blockers
Depolarizing nicotinic neuromuscular blocker
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Succinylcholine
Depolarizing neuromuscular blocker
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Non-depolarizing NMJ blockers
Non-depolarizing nicotinic neuromuscular blockers
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Tubocurarine
Non-depolarizing neuromuscular blocker
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Pancuronium
Non-depolarizing neuromuscular blocker
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Rocuronium
Non-depolarizing neuromuscular blocker
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Mivacurium
Non-depolarizing neuromuscular blocker