Targeted Therapy Classes

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Last updated 12:33 PM on 6/9/26
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44 Terms

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Antibody Inhibitors of EGFRs

Cetuximab

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Antibody Inhibitors of EGFRs

Panitumumab

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Antibody Inhibitors of EGFRs

Necitumumab

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1st Gen Tyrosine Kinase Inhibitors (TKIs) of EGFR

Gefitinib

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1st Gen Tyrosine Kinase Inhibitors (TKIs) of EGFR

Erlotinib

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2nd Gen Tyrosine Kinase Inhibitors (TKIs) of EGFR

Afatinib

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2nd Gen Tyrosine Kinase Inhibitors (TKIs) of EGFR

Neratinib

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3rd Gen Tyrosine Kinase Inhibitors (TKIs) of EGFR

Osimertinib

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3rd Gen Tyrosine Kinase Inhibitors (TKIs) of EGFR

Avitinib

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Antibody Inhibitors of HER2/Neu

Trastuzumab

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Antibody Inhibitors of HER2/Neu

Pertuzumab

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Protein Tyrosine Kinase Inhibitors of HER2/Neu

Lapatinib

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Protein Tyrosine Kinase Inhibitors of HER2/Neu

Neratinib

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RAF Kinase Inhibitors

Vemurafenib

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RAF Kinase Inhibitors

Dabrafenib

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MEK Kinase Inhibitors

Trametinib

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MEK Kinase Inhibitors

Cobimetanib

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BCR-ABL Kinase Inhibitors

Imatinib

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BCR-ABL Kinase Inhibitors

Dasatinib

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BCR-ABL Kinase Inhibitors

Nilotinib

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BCR-ABL Kinase Inhibitors

Ponatinib

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mTOR Inhibitors

Rapamycin (Sirolimus)

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mTOR Inhibitors

Everolimus

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mTOR Inhibitors

Temsirolimus

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Cyclin-Dependent Kinase (CDK4/6) Inhibitors

Palbociclib

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Angiogenesis Inhibitors Antibodies

Bevacizumab

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Angiogenesis Inhibitors Antibodies

Ranibizumab

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Angiogenesis Inhibitors Antibodies

Ramucirumab

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Small Molecule Kinase Angiogenesis Inhibitors

Sunitinib

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Small Molecule Kinase Angiogenesis Inhibitors

Sorafenib

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Small Molecule Kinase Angiogenesis Inhibitors

Pazopanib

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PD-1 Inhibitors

Nivolumab

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PD-1 Inhibitors

Pembrolizumab

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PD-L1 Inhibitors

Atezolimumab

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CTLA-4 Inhibitors

Ipilimumab

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Anti-CD20 Antibody

Rituximab

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Proteasome Inhibitors

Bortezomib

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Proteasome Inhibitors

Carfilzomib

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Proteasome Inhibitors

Ixazomib

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Enzyme to break down toxic methotrexate metabolites

Glucarpidase

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Rescue agent for methotrexate toxicity

Leucovorin

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Cytoprotective agent used prior to radiation or alkylating agents

Amifostine

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Cardioprotective agent used with anthracyclines

Dexrazoxane

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Antidote to prevent acrolein-induced bladder toxicity

MESNA