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+ H2O


+ R’OH


+ R’-NH2


+ R’COOH


+ (1) R’MgX
(2) H2O


+ R2’CuLi


+ (1) NaBH4 or LiAlH4
(2) H2O


+ LiAlH(O-t-Bu)3




+ H2O


+ R’OH/ H+


+ R’NH2














+ H2O/H+ or -OH


+ R'“OH/H+ or -OR”


+ R”NH2


+ (1) LiAlH4/(2) H2O


+ (1) 2R”MgX/ (2) H2O


+ (1) DIBAL-H -78°C/(2) H2O












+ H2O/H+ or -OH


+ POCl3/(or P2O5)




