Biotherapy Nomeclature

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Last updated 7:31 PM on 4/21/26
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41 Terms

1
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Small-Molecular Targeted Therapy Format

Prefix + substem(s) + stem

2
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Small-Molecular Targeted Therapy stem

-ib (except HDAC and BCL-2)

3
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-tini-

Tyrosine kinase inhibitors

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afatinib

Tyrosine kinase inhibitor

5
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Axitinib

Tyrosine kinase inhibitor

6
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Bosutinib

Tyrosine kinase inhibitor

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Dasatinib

Tyrosine kinase inhibitor

8
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Erlotinib

Tyrosine kinase inhibitor

9
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Gefitinib

Tyrosine kinase inhibitor

10
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Sunitinib

Tyrosine kinase inhibitor

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-rafe-

RAF tyrosine kinase RAF/RAS/MEK pathway

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Dabrafenib

RAF tyrosine kinase RAF/RAS/MEK pathway

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Regorafinib

RAF tyrosine kinase RAF/RAS/MEK pathway

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Sorafenib

RAF tyrosine kinase RAF/RAS/MEK pathway

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Vemurafenib

RAF tyrosine kinase RAF/RAS/MEK pathway

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-metin-

MEK tyrosine kinase RAF/RAS/MEK pathway

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Cobimetinib

MEK tyrosine kinase RAF/RAS/MEK pathway

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Trametinib

MEK tyrosine kinase RAF/RAS/MEK pathway

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-den-

IDH2 enzyme inhibitor

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Enasidenib

IDH2 enzyme inhibitor

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-par-

PARP inhibitors

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Olaparib

PARP inhibitors

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Rucaparib

PARP inhibitors

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-Lis-

PI3K

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Idelalisib

PI3K

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-deg-

Sonic hedgehog pathway inhibitors

27
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Sonidegib

Sonic hedgehog pathway inhibitors

28
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Vismodegib

Sonic hedgehog pathway inhibitors

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-cicl-

CDK 4 & 6

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Palbociclib

CDK 4 & 6

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-zo-

Proteasome inhibitors

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Bortezomib

Proteasome inhibitors

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Carfilzomib

Proteasome inhibitors

34
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Ixazomib

Proteasome inhibitors

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-inostat

HDAC

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Vorinostate

HDAC

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Belinostat

HDAC

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Panobinostat

HDAC

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-toclax

BCL-2 inhibitors

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Venetoclax

BCL-2 inhibitors

41
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