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Opioid Analgesics
Strong pain-relief medication
Work by attaching to opioid receptors in the brain + spinal cord, which blocks pain signals
Used for moderate to severe pain
Must be used carefully and exactly as prescribed because they can cause dependence, drowsiness, and slowed breathing
Tramadol
Trade Name: Vitram, Vitracet; Classification: Opioid analgesic (synthetic), SNRI-like activity; Indication: Moderate Pain; Notes: Schedule IV, low risk for dependence and misuse
Codeine
Trade Name: Codeine; Classification: Opioid analgesic; Indication: Mild to Moderate Pain; Notes: Schedule II, schedule III-IV in combination. For pain as a cough suppressant. Found in combination with acetaminophen. Less potent than both hydrocodone + oxycodone.
Hydrocodone
Trade Name: Vicodin, Norco; Classification: Opioid analgesic; Indication: Moderate to Severe Pain; Notes: Schedule II. Found in combination with acetaminophen. Slightly less potent than oxycodone. High risk for dependence + abuse.
Oxycodone
Trade Name: Oxycontin, Percocet; Classification: Opioid analgesic; Indication: Moderate to Severe Pain; Notes: Schedule II. Found in combination with acetaminophen. Oxycontin is long-acting. High risk for dependence + abuse.
Meperidine
Trade Name: Demerol; Classification: Opioid analgesic; Indication: Moderate to Severe Pain; Notes: Schedule II. Less common due to potential for toxic metabolite accumulation which can cause seizures.
Oxymorphone
Trade Name: Opana; Classification: Opioid analgesic; Indication: Moderate to Severe Pain; Notes: Schedule II. High potency. High risk for dependence + abuse.
Morphine
Trade Name: Morphine; Classification: Opioid analgesic; Indication: Severe Pain; Notes: Schedule II. Available in many forms (oral, IV). High risk for dependence.
Fentanyl
Trade Name: Duragesic, Sublimaze; Classification: Opioid analgesic, Semi-Synthetic; Indication: Severe Pain; Notes: Schedule II. Often used in transdermal patches or IV. High risk of overdose and dependence. Extremely potent; even small variations in dose can be fatal.
Hydromorphone
Trade Name: Dilaudid; Classification: Opioid analgesic; Indication: Severe Pain; Notes: Schedule I. Very potent. High risk of dependence and abuse.
Methadone
Trade Name: Methadone, Dolophine; Classification: Opioid analgesic; Indication: Chronic Pain; Notes: Schedule I. Long Acting, used for chronic pain opioid dependence. Methadone has a very long half-life, requires specialized titration, careful monitoring.
Tylenol with Codeine; Tylenol #3, #4 (Combination Medication)
Acetaminophen-codeine
Lorcet, Lortab, Norco, Vicodin (Combination Medication)
Hydrocodone-acetaminophen
Endocet, Percocet (Combination Medication)
Oxycodone-acetaminophen
Endodan, Percodan (Combination Medication)
Oxycodone-aspirin
Cambunox (Combination Medication)
Oxycodone-ibuprofen
Talwin NX (Combination Medication)
Pentazocine-naloxone