EXAM 2 Drugs

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Cholinergic Drugs (Direct and Indirect)
Bethancol, Pilocarpine
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Bethancol
Urecholine - Direct cholinergic agonist that activates muscarinic receptors.
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Pilocarpine
Isopto, Carpine - Direct cholinergic agonist that activates muscarinic receptors.
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Donezepil
Aricept - Acetylcholinesterase inhibitor that increases the availability of acetylcholine in the brain.
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Neostigmine
Prostigmin - Acetylcholinesterase inhibitor that increases the availability of acetylcholine at the neuromuscular junction.
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Physostigmine
Antilirium - Acetylcholinesterase inhibitor that increases the availability of acetylcholine in the central nervous system.
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Pyridostigmine
Mestinon, Regonol - Acetylcholinesterase inhibitor that increases the availability of acetylcholine at the neuromuscular junction.
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Rivastigmine
Exelon - Acetylcholinesterase inhibitor that increases the availability of acetylcholine in the brain.
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Anticholinergics
Atropine, Benztropine, Ipratropium, Oxybutinin, Propantheline, Scopolamine
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Atropine
AtroPen - Blocks muscarinic receptors.
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Benztropine
Cogentin - Blocks muscarinic receptors.
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Ipratropium
Atrovent - Blocks muscarinic receptors.
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Oxybutynin
Ditropan, Oxytrol - Blocks muscarinic receptors.
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Propantheline
Pro-Banthne - Blocks muscarinic receptors.
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Scopolamine
Transderm-Scop - Blocks muscarinic receptors.
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Adrenergic Drugs
Albuterol, Dpotamine, Epinetphrine, Isoprotenernol, Norepinephrine, Phenylephrine, Pseudoephedrine
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Albuterol
Proventil, Ventolin - Selective beta-2 adrenergic agonist.
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Dopamine
Dopastat - Dopamine receptor agonist.
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Epinephrine
Adrenaline - Non-selective adrenergic agonist
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Isoproterenol
Isuprel - Non-selective beta adrenergic agonist
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Norepinephrine
Leviphed - Non-selective adrenergic agonist
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Phenylephrine
Neo-synephrine - Alpha-1 adrenergic agonist
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Pseudoephedrine
Sudafed - Non-selective adrenergic agonist
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Anti-Andrenergic Drugs
Atenolol, Bisoprolol, Cartelol, Carvedilol, Metoprolol, Prazosin, Propanolol, Tamsulosin
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Atenolol
Tenormin - Selective beta-1 adrenergic receptor antagonist
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Bisoprolol
Zebeta - Selective beta-1 adrenergic receptor antagonist
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Cartelol
Cartrol - Non-selective beta adrenergic receptor antagonist
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Carvedilol
Coreg - Non-selective beta adrenergic receptor antagonist and alpha-1 adrenergic receptor antagonist
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Metoprolol
Lopressor, Torpol - Selective beta-1 adrenergic receptor antagonist
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Prazosin
Minipress - Alpha-1 adrenergic receptor antagonist
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Propanolol
Inderal- Non-selective beta adrenergic receptor antagonist
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Tamsulosin
Flomax - Alpha-1 adrenergic receptor antagonist
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Antidepressants
Escitalopram, fluoxetine, sertraline, duloxetine, bupropion, imipramine, trimipramine, phenelzine
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Escitalopram
lexapro - SSRI
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fluoxetine
prozac - SSRI
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sertraline
zoloft - SSRI
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duloxetine
cymbalta - SNRI
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bupropion
wellbutrin
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imipramine
tofranil - SNRI
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trimipramine
surmontil - SNRI
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phenelzine
nardil - MAOI
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beznzodiazepines
alprazolam, diazepam, lorazepam
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aprazolam
xanax
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diazepam
valium
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lorazepam
ativan
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barbituates
pentobarbital, butabarbital, phenobarbital
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pentobarbital
nembutal
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butabarbital
butabarbital
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phenobarbital
luminal
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nonbenzodiazepines, non barbituate CNS depressants
eszopiclone, zaleplon, zolpidem
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eszopiclone
lunesta
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zaleplon
sonata
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zolpidem
ambien
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orexin receptor blocker
suvorexant
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suvorexant
belsomra - orexin receptor antagonist
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melatonin receptor agonists
ramelteon - melatonin receptor agonist
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ramelteon
rozerem
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Propranolol
Inderal
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Atenolol
Tenormin
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Beta blockers used in anxiety/insomnia
propranolol and atenolol
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Gaba potentiating drugs
gabapentin, pregabalin, topiramate
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gabapentin
gralise
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pregabalin
lyrica
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topiramate
topomax
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hydantoins
phenytoin
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phenytoin
dilantin
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phenytoin-related drugs
carbamazepine, valproic acid
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carbamazepine
tegretol
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valproic acid
depakene
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succinimides
ethosuximide
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ethosuximide
zaronitin
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mood stabilizers
lithium
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lithium
eskalith
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atypical antipsychotic drugs
aripiprazole, risperiidone, clozapine
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aripiprazole
abilify
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risperiidone
risperdal
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clozapine
clozaril
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CNS stimulants
D/L amphetamine, methylphenidate
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D/L amphetamine
adderall
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methylphenidate
ritalin
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ADHD nonstimulant drugs
atomoxetine
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atomoxetine
strattera
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phenothiazines
chlorpromazine, prochlorperazine
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prochloperazine
compazine
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nonphenothiazines
haloperidol
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haloperidol
haldol
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opiod agonists
fentanyl, morphine, codeine, hydrocodone, oxycodone
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hydrocodone
hycodan
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oxycodone
oxycontin
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opiod antagonists
nalaxone
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nalaxone
narcan, evzio
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opiod w mixed agonist/antagonist effects
buprenorphine
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buprenorphine
buprenex
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NSAIDS
aspirin, ibuprofen, indomethacin, naproxen
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ibuprofen
advil, motrin
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indomethacin
indocin
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naproxen
aleve (sodium form), naprelan
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cox-2 selective inhibitors
celexoxib
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celexoxib
celebrex
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centrally acting analgesics
acetaminophen, tramadol