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bupropion
(Wellbutrin, Zyban)
norepinephrine-dopamine reuptake inhibitors (NDRIs)
Depression, SAD, Smoking Cessation
(IR) 100mg po bid x 3 days, the increase to 150mg po bid
(ER) 150mg po daily, titrate up to 300mg
Agitation, constipation, dizziness, headache, insomnia
Avoid alcohol, take at the same time each day.
varenicline
(Chantix)
Smoking Cessation (nicotinic receptor partial agonist)
Smoking Cessation
0.5mg po daily x 3 days, then bid x 4 days, then 1mg po bid for 4-6 weeks
Dream disorder, nausea, headache, insomnia, irritabilityย
Take drug after eating and with a full glass of water. Contact HCP if there is onset of mental/sleep issues.
warfarin
(Coumadin)
Anticoagulants
Atrial Fibrillation, risk of MI
2-5mg po daily, adjust dose based on INR.
Bleeding, anemia, epistaxis, rash, hemorrhage
Report signs of hemorrhage, tissue necrosis. Avoid situations where you could bruise or get cut.
apixaban
(Eliquis)
Anticoagulants
Atrial Fibrillation, risk of DVT
5mg po bid
Bleeding, elevated LFTs, nausea, hypotension
Seek medical attention if any unexpected bleeding or trouble breathing.
rivaroxaban
(Xarelto)
Anticoagulants
Risk of thromboembolism, treatment of DVT/PE, coronary heart disease
2.5mg-15mg po bid
Bleeding, cough, peripheral edema, dizziness, headache
Educate patient of signs and symptoms of bleeding and interactions w/ other anticoagulant/antiplatelet medications.
clopidogrel
(Plavix)
Anticoagulants
MI, Thrombosis prevention
75mg po daily
Headache, arthralgia, backache, epistaxis, gastritisย
Report signs/symptoms of bleeding, do not stop abruptly.
albuterol AND levalbuterol
(Ventolin or ProAir and Xopenex)
(Asthma/COPD (PRN))
(SABA)
(1-2 puffs q 4-6 hrs prn.)
(Side Effects: Tremor, nervousness, nausea, throat irritation, tachycardia.)
(Counseling Points: Device Use Counseling)
Fluticasone
(Flovent)
(Asthma/COPD (Maintenance))
(Corticosteroids)
1 puff bid for chronic asthma treatment. Titrate up as prescribed.
(Side Effects: Candidiasis, Fatigue, Headache, Arthralgia)
Counseling Points: Rinse mouth, inhaler instructions
Budesonide
(Pulmicort)
Asthma/COPD (Manage Symptoms)
Corticosteroids
Dry Inhaler: 2 puffs bid, up to 4 puffs bid.
Nebulizer: 0.5-1mg in 1-2 divided doses daily.
Side Effects: Cough, headache, respiratory tract infection, ear infection, rhinitis
Counseling Points: Swirl suspension before use, proper inhalation technique.
Fluticasone/Salmeterol
(Advair)
Asthma/COPD (Manage symptoms)
Corticosteroid/LABA
2 MDI puffs/1 disk puff q 12 hours prn asthma.
Side Effects: Headache, pharyngitis, nausea, upper respiratory tract infection, difficulty speaking
Counseling Points: Proper Inhaler technique and mouth rinsing.
Budesonide/Formoterol
(Symbicort)
Asthma/COPD (Manage Symptoms)
Corticosteroid/LABA
Asthma: 2 puffs bid, can titrate up.
COPD: 2 puffs bid of high conc. solution.
Side Effects: Respiratory tract infections, headache, cough
Counseling Points: Proper inhalation technique and mouth rinsing.
Fluticasone/vilanterol
(Breo Ellipta)
COPD/Asthma (Manage symptoms)
Corticosteroid/LABA
1 puff qd
Side Effects: Candidiasis, osteoporosis, increased risk of infection
Counseling Points: Risks, mouth rinsing, inhalation technique
Ipratropium/albuterol
(Combivent)
COPD/Asthma
Anticholinergic/Beta-2 Agonist
1 puff qd or 3mL nebulizer q6h.
Side Effects: Bronchitis, upper respiratory tract infection, nausea, tachycardia
Counseling Points: Instruct on proper inhalation technique and cleaning. Use entire vial of nebulizer solution at once to avoid contamination.
Tiotropium
(Spiriva)
COPD/Asthma (Maintenance)
Anticholinergic
COPD: Inhale 1 capsule or 2 puffs of solution once daily.
Asthma: 2 actuations of aerosol solution once daily.
Side Effects: Dry mouth, upper respiratory tract infection, headache, constipation
Instruct proper use of inhalation device, remind that this is not indicated for acute bronchospasm.
umeclidinium/vilanterol
(Anoro Ellipta)
COPD (Maintenance)
Anticholinergic/Beta-2 Agonist
1 puff qd
Side Effects: Rhinitis, respiratory tract infections, muscle spasms, cough, joint pain
Instruct on proper inhaler use and mouth rinsing.
umeclidinium/vilanterol/fluticasone
(Trelegy)
COPD/Asthma (Maintenance)
Anticholinergic/Beta-2 Agonist/Corticosteroid
1 puff qd
Side Effects: Candidiasis, upper respiratory tract infections, cough, headache, joint pain
Instruct on proper inhaler use and mouth rinsing.
Prednisone AND Methylprednisolone
(Deltasone and Medrol)
Inflammatory conditions like dermatitis and bronchitis, severe allergies.
Corticosteroids (oral)
(5-60mg/4-64) po daily titrating the dose down with/without dosepak as prescribed.
Side Effects: GI Upset, impaired skin healing, euphoria, hypertension, immunosuppression
Take with meals to prevent GI upset. Inform on incidence of long-term effects if being used long-term.
Montelukast
(Singulair)
Asthma, exercise-induced bronchoconstriction, seasonal congestion
Leukotriene Receptor Antagonist (oral)
Children: 5mg po daily
Adults: 10mg po daily
Side Effects: Dizziness, fatigue, nausea, rash, rare neurological problems (depression).
Counsel on long-term use and incidence of rare neurological effects.
Lisinopril
(Zestril, Prinivil)
ACE inhibitors
Hypertension, heart failure, arrhythmia
2.5-10mg po daily
Dizziness, hypotension, dry cough, swelling of face
Use potassium or salt substitutes only under medical supervision.
Enalapril
(Vasotec)
ACE inhibitors
Hypertension, heart failure
2.5-10mg po daily
High serum creatinine (reduced kidney function), dizziness, hypotension, swelling of face
Use caution when getting up from a seated/lying position. Avoid pregnancy.
benazepril
(Lotensin)
ACE inhibitors
Hypertension
10mg po daily
Rare: Constipation, facial swelling, dizziness, cough
Avoid pregnancy, may cause dizziness, caution using salt substitutes.
Losartan
(Cozaar)
Angiotensin Receptor Blockers
(ARBs)
Hypertension, stroke chance reduction, diabetic management
25-50 mg po daily
Headache, back pain, anorexia, constipation, dizziness
Avoid sudden discontinuation, use salt subs under supervision.
Valsartan
(Diovan)
Angiotensin Receptor Blockers
(ARBs)
Hypertension, heart failure
HTN: 80-160mg po daily
Heart Failure: 20-40mg po bid
Dizziness, increased blood urea nitrogen (BUN) levels, back pain, cough
Avoid sudden discontinuation, salt subs only under supervision.
Olmesartan
(Benicar)
Angiotensin Receptor Blockers
(ARBs)
HTN
20-40mg po daily
Rarely: Back pain, dizziness, headache, hyperkalemia
Use salt subs under supervision, may cause dizziness, avoid pregnancy.
Sacubitril/Valsartan
(Entresto)
Neprilysin Inhibitor + ARB
Heart Failure
24mg/36mg po bid (or other available dose amount)
Hypotension, hyperkalemia, increased serum creatinine, dizziness
Do not discontinue abruptly, use salt substitutes under supervision
Canagliflozin
(Invokana)
SGLT-2 inhibitors
Diabetes mellitus
100-300mg po daily before first meal (if albumin excretion is >300mg/d)
GU fungal infection, hypoglycemia, hyperkalemia
Take before first meal of the day to reduce post-meal hyperglycemia. Be aware of ulcer symptoms.
Dapagliflozin
(Farxiga)
SGLT-2 inhibitors
Diabetes mellitus, heart failure, kidney disease
5-10mg po daily
GU fungal infection, hypoglycemia, hypovolemia, UTIs
Take before first meal of the day to reduce post-meal hyperglycemia.
Amlodipine
(Norvasc)
Calcium Channel Blockers
HTN, Angina
5-10mg po daily
Peripheral edema, abdominal pain, arthralgia, dizziness, fatigue
Report symptoms of hypotension, avoid drinking alcohol.
Diltiazem
(Cardizem, Dilacor, Tiazac)
Calciumย Channel Blockers
HTN, Angina
60-120mg (ER) po bid, for angina 30mg (IR) po qid
Edema, bradycardia, constipation, dizziness
Report symptomatic hypotension and edema. Multiple brand names/properties of drug.
Nifedepine
(Procardia, Adalat)
Calciumย Channel Blockers
HTN, Angina
30-60mg po daily (ER)
Flushing, headache, dizziness, weakness, nausea
Take Adalat CC on an empty stomach, monitor hypotension and edema symptoms.
Verapamil
(Calan, Verelan)
Calciumย Channel Blockers
Angina, arrhythmia, HTN
80-120 mg po tid (IR)
Gingival hyperplasia, bradyarrhythmia, constipation, dizziness
Do not crush or chew ER products, ER capsule products may be sprinkled on food and swallowed.
Atenolol
(Tenormin)
Beta Blockers
Angina, HTN, heart attack (AMI)
25-50mg po daily, may titrate up
Bradyarrhythmias, cold extremities, dizziness, fatigue, hypotension
Take on an empty stomach, avoid abrupt discontinuation
Metoprolol Succinate
(Toprol XL)
Beta Blockers
Angina, Heart Failure, HTN
100mg ER po or 25-100mg ER bid.
Dizziness, fatigue, hypotension, arthralgia
Avoid alcohol and abruptly stopping the medication.
Metoprolol tartrate
(Lopressor)
Beta Blockers
Angina, HTN, AMI
25-50mg po bid or q6h prn AMI
Dizziness, fatigue, hypotension, arthralgia
Take on empty stomach, avoid alcohol and stopping abruptly.
Labetalol
(Normodyne)
Beta Blockers
HTN
100mg po bid
Dizziness, nausea, hypotension, bradyarrhythmias
Report signs of hypotension, avoid alcohol.
Carvedilol
(Coreg)
Beta Blockers
Heart Failure, HTN
3.125-6.25mg po bid
Cold extremities, dizziness, diarrhea, fatigue, hypotension
Take with food/milk, report symptoms of heart failure.
Propranolol
(Inderal)
Beta Blocker
Angina, HTN, dysrhythmia
80-320mg po daily, HTN and dysrhythmia will usually split into 2 doses.
Hypotension, bradyarrhythmias, bronchospasm, constipation
Take on an empty stomach (IR). Avoid alcohol.
Hydrochlorothiazide (HCTZ)
(Hydrodiuril)
Thiazide Diuretic
Edema, HTN
12.5-25mg po daily, double for Edema
Hypotension, dizziness, headache, constipation
Take early in the morning to avoid nocturia.
Chlorthalidone
(Hygroton, Thalitone)
Thiazide Diuertic
HTN, Edema
12.5-25mg po daily
Dizziness, hypotension, hyperuricemia, anorexia
Take in the morning with food. Report signs of dyspnea, hypotension.
Furosemide
(Lasix)
Loop Diuretics
Edema due to heart/renal failure
20-80mg po daily
Hyperuricemia, constipation, headache, hyperglycemia
Avoid alcohol and NSAIDs, increased sun sensitivity.
Spironolactone
(Aldactone)
Potassium sparing diuretic
Heart Failure, Aldosteronism, HTN, liver cirrhosis
12.5-25mg po daily, titrated up for liver cirrhosis
Breast tenderness, diarrhea, menstruation disorders, gastritis
Avoid driving, may cause dizziness.
Lovastatin
(Mevacor)
HMG-CoA Reductase inhibitors (Statins)
Arteriosclerosis, hypercholesterolemia
10-80mg po daily
Increased creatinine phosphokinase, infection, abdominal pain, constipation
Take IR with evening meal, take ER at bedtime. Avoid alcohol/grapefruit juice.
Atorvastatin
(Lipitor)
HMG-CoA Reductase Inhibitors (Statins)
Atherosclerosis, cardiovascular event prevention, high cholesterol
10-80mg po daily
Myopathy, diarrhea, headache, nasopharyngitis, increased liver enzymes
Avoid alcohol/grapefruit juice.
Simvastatin
(Zocor)
HMG-CoA Reductase inhibitors (Statins)
Hyperlipidemia, atherosclerosis, high cholesterol
20-40mg po daily
Abdominal pain, constipation, diarrhea, headache, increased liver enzymes
Avoid alcohol, consult HCP before starting new medications/supplements.
Pravastatin
(Pravachol)
HMG-CoA Reductase Inhibitors (Statins)
Stroke prevention, high cholesterol, hyperlipidemia
40-80mg po daily
Musculoskeletal pain, upper respiratory tract infection, headache, heartburn
Take in evening, avoid alcohol.
Rosuvastatin
(Crestor)
HMG-CoA Reductase Inhibitor (Statins)
Hyperlipidemia, high cholesterol
5-40mg po daily
Arthralgia, abdominal pain, fatigue, constipation
Avoid alcohol.
Gemfibrozil
(Lopid)
Fibrates
Arteriosclerosis, hyperlipoproteinemia
600mg po bid
Indigestion, abdominal pain, atrial fibrillation, constipation
Monitor symptoms of rhabdomyolysis, yellowing of skin.
Fenofibrate
(Tricor, Lofibra)
Fibrates
Hypertriglyceridemia, hyperlipidemia
35-200mg po daily
Hyperhomocysteinemia, abdominal pain, constipation, diarrhea
Tk 1 hr before or 4-6hrs after bile acid binding resin.
Ezetimibe
(Zetia)
Cholesterol absorption inhibitor
High cholesterol, hyperlipidemia, sitosterolemia
10mg po daily
Abdominal pain, constipation, diarrhea, headache
Tk 2h before or 4h after bile acid binding resin.