Drug Target and Type

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Last updated 6:56 PM on 10/1/26
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18 Terms

1
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Salbutamol

B2 receptors on bronchial smooth muscle

Agonist

2
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Nifedipine

L-type VG Ca channels

Ca channel blocker/Gating Inhibitor/Antagonist

3
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Enalapril

ACE

Competitive inhibitor

4
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Simvastatin

HMG-CoA Reductase

Competitive Inhibitor

5
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Aspirin

Cyclooxygenase

Irreversible competitive inhibitor

6
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Metformin

7
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Fluoxetine

5HT (2A, 2C, 6 & 2B)

Antagonist (competitive)

8
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Imatinib

Bcr-Abl TK receptor

Competitive Inhibitor

9
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Fentanyl

mu Opioid Receptor

Agonist

10
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Metoprolol

B1 receptors

Antagonist (competitive)

11
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Furosemide

Na/K/Cl Symporter

Competitive inhibitor

12
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Sildenafil

PDE5

Competitive Inhibitor

13
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Clopidogrel

P2Y12

Antagonist (non-competitive, irreversible)

14
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Prednisolone

Glucocorticoid Receptor

Agonist

15
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Ranitidine

H2 receptor

Antagonist (competitive)

16
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Vancomycin

NAM and NAG (D-Ala-D-Ala)

Inhibitor

17
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Rituximab

CD20 Antigen (on B cells)

Monoclonal Antibody

18
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Diazepam

GABA A

Positive Allosteric Modulator