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Chapter 17
Phenylephrine
A1 agonist
Sympathomimetic
Dilates eyes
Beta blockers
Sympatholytic
Pilocarpine
Muscarinic agonist
Parasympathomimetic
Pupil constriction
Atropine
Muscarinic antagonist
Anticholinergic (Blocks ACh)
Higher heart rate
Alpha-1 receptor
Releases intracellular Ca2+
Alpha-2 receptor
Decreases cAMP
Beta-1 receptor
Increases cAMP; more heart stimuli
Beta-2 receptor
Increases cAMP; Relaxes lungs
Beta-3 receptor
increases cAMP; breaks down fat
Tropicamide
Muscarinic antagonist
Pupil dilation
Scopolamine
Muscarinic antagonist
Motion sickness