- AD is characterized by degeneration of cholinergic neurons leading to deficiencies in ACh
- Medications to treat AD are acetylcholinesterase (AChE) inhibitors
- Inhibits the breakdown of ACH
- Increases ACh levels in the neuron receptors
- AChE inhibitors increase cognitive function for mild to moderate AD patients
- Are classified into reversible and nonreversible AChE inhibitors
Rivastigmine
- Used for mild to moderate AD
- Increases the amount of ACh at cholinergic synapses
- It is absorbed faster through the GI ***without*** food
- Contraindicated in patients with liver and renal dysfunction