Metabolism & Nutrient Fate
- Definition & Scope
- Collective term for all chemical reactions sustaining life
- Mathematically expressed as: \text{Metabolism}=\text{Catabolism}+\text{Anabolism}
- Constant balance between energy release (to power work/heat) and energy investment (to build/repair)
- Big-picture Significance
- Links nutrition, endocrinology, physiology & cellular biology
- Malfunction → diabetes, obesity, cachexia, inborn errors of metabolism
- Practical/ethical lens: informs public-health policy, food security, sustainable agriculture
Fate of Digested Nutrients
- Immediate Energy
- Oxidised in catabolic pathways → ATP + heat
- Drives muscular contraction, ion pumps, active transport, biosynthesis
- Raw Material for Biosynthesis
- Precursors for new macromolecules (proteins, nucleic acids, polysaccharides, lipids)
- Vital for growth, repair & immune competence
- Storage Pathways
- Glycogenesis → glycogen (liver, skeletal muscle)
- Lipogenesis → triglycerides (adipocytes, liver)
- Protein accretion in lean tissues
Reaction Types
- Catabolic Reactions
- Break chemical bonds; large → small molecules
- Net \Delta G<0, releasing energy (often captured as ATP, NADH, FADH$_2$)
- Examples: glycolysis, β-oxidation, proteolysis
- Anabolic Reactions
- Form chemical bonds; small → large molecules
- Require energy input (usually from ATP/NADPH)
- Examples: glycogen synthesis, fatty-acid synthase, ribosomal protein synthesis
Cellular Energy Currency
- Goal: Convert nutrient energy into a format used by nearly every enzyme system
- Energy Source: Macromolecule oxidation (mainly glucose & triglycerides)
- Currency: ATP, augmented by GTP, UTP, CTP for specialized reactions
ATP: Structure & Function
- Diagrammatic Features
- Adenine (nitrogenous base) + ribose ⇒ adenosine
- Three phosphate groups linked by two high-energy phosphoanhydride bonds
- Hydrolysis: \text{ATP}+\text{H}2\text{O} \rightarrow \text{ADP}+\text{P}i+\text{Energy} (≈ 7.3 \text{ kcal·mol}^{-1} under standard conditions)
- Role Shuttling Energy
- Catabolism → synthesises ATP
- Anabolism/transport → splits ATP, harnessing energy
- Recycling Rate: Entire body pool (~50–75 g) turned over every minute at rest
Review of Major Biological Macromolecules
- Carbohydrates
- Monomer: glucose
- Polymers: amylose & amylopectin (starch), glycogen, cellulose (fiber)
- Key bond: glycosidic linkage (\alpha or \beta)
- Nucleic Acids
- Pentose (ribose or deoxyribose) + phosphate + nitrogenous base (purine/pyrimidine)
- Phosphodiester bonds; bases A, G (purines) & C, T, U (pyrimidines)
- Proteins
- Built from 20 amino acids via peptide bonds
- Levels: primary → secondary (\alpha-helix/\beta-sheet) → tertiary → quaternary (e.g. hemoglobin)
- Lipids
- Triglyceride = glycerol + 3 fatty acids
- Also phospholipids, cholesterol, steroid hormones, myelin
Preferred ATP Energy Sources
- Priority Hierarchy
- 1st: glucose & triglycerides
- Brain & erythrocytes: require glucose (brain can use ketone bodies after prolonged fasting)
- Other tissues switch flexibly between lipids & glucose
- Last-resort: amino acids (protein catabolism)
- Physiological Set-point: Blood glucose maintained ≈ 70\text{–}100\,\text{mg·dL}^{-1}
Inter-Conversion Pathways
- Producing Glucose (Gluconeogenesis)
- Substrates: lactate, pyruvate, certain glucogenic amino acids
- Location: liver (90 %), kidney cortex (10 %)
- From Glucose
- Glycogenesis (short-term storage)
- Lipogenesis (excess → triglycerides)
- Insulin
- Released when blood glucose↑
- Actions: ↑ cellular glucose uptake; ↑ glycogen & lipid synthesis; ↓ glucagon secretion
- Glucagon
- Trigger: blood glucose↓, amino acids↑
- Actions: ↑ hepatic gluconeogenesis & glycogenolysis; ↑ lipolysis; ↓ insulin
- Cortisol
- Released under stress/circadian drive
- Mobilises fuel: ↑ gluconeogenesis, protein catabolism; anti-insulin effects
- Growth Hormone + IGF-1
- Stimuli: sleep, exercise, high-protein meal, hypoglycaemia, trauma
- Effects: ↑ protein synthesis (esp. muscle), bone growth, lipolysis
Measuring Energy Intake/Expenditure
- Calorie Conventions
- 1\,\text{cal} (chemistry) = heat to raise 1\,\text{g H}_2\text{O} by 1^{\circ}\text{C}
- 1\,\text{Calorie}=1\,\text{kcal}=1000\,\text{cal}
- Macronutrient Energy Density
- Carbohydrate: \approx4\,\text{kcal·g}^{-1}
- Protein: \approx4\,\text{kcal·g}^{-1}
- Lipid: \approx9\,\text{kcal·g}^{-1}
- Practical Note: Food labels use “Calories” (kcal); accurate tracking informs weight management & metabolic research
- Dietary Fiber
- Non-digestible polysaccharides
- Water-soluble (e.g. pectins) → modulate cholesterol/glucose absorption
- Insoluble (e.g. cellulose) → bowel motility, microbiome substrate
- Other Roles
- Ribose ↑ nucleotide synthesis (e.g. ATP, DNA/RNA)
- Glycoproteins & glycolipids in cell-cell recognition (immune & developmental biology)
Lipids: Non-Fuel Functions
- Membrane Architecture: phospholipid bilayer integrity & fluidity
- Cholesterol Derivatives: steroid hormones, bile salts, vitamin D
- Cell Signalling: eicosanoids, phosphatidylinositol cascade
- Myelin: electrical insulation of neurons
- Functional Diversity
- Structure (collagen, cytoskeleton, muscle), enzymes, antibodies, hormones, transport proteins (albumin, hemoglobin)
- Nitrogen Disposal
- Catabolism liberates NH$_3$ (toxic)
- Urea Cycle (liver): converts NH$3$ + CO$2$ → urea → excreted in urine
- Failure → hyperammonaemia (neurological damage)
Micronutrients
- Vitamins
- Water-soluble: B-complex (B$1$–B${12}$), C
- Fat-soluble: A, D, E, K
- Minerals
- Major (>100 mg·day$^{-1}$): Na, K, Ca, P, Mg, Cl
- Trace: Fe, Cu, Zn, I, S, Mn, Co, F, Se, Cr, Mo
- Metabolic Co-factors: many serve as enzyme prosthetic groups (e.g. Fe in cytochromes, Zn in DNA-binding proteins)
Essential Nutrients
- Cannot be Synthesised in Adequate Quantities
- Fatty Acids: linoleic (ω-6), α-linolenic (ω-3); possibly arachidonic (conditional)
- Amino Acids: 9 indispensable (His, Ile, Leu, Lys, Met, Phe, Thr, Trp, Val) + 6 conditionally essential in infants/illness
- Vitamins: most, except some vitamin D (skin) & K (gut flora)
- Minerals: all must be ingested
- Dietary Planning Implication: variety of whole foods ensures sufficiency; vegan/vegetarian diets require B$_{12}$ monitoring
Integrative & Ethical/Philosophical Connections
- Systems Perspective: Hormonal orchestration exemplifies homeostasis — dynamic stability despite fluctuating intake/needs
- Public Health: Understanding metabolism guides interventions against metabolic syndrome & malnutrition
- Environmental Ethics: Choosing nutrient-dense, sustainably produced foods reduces ecological footprint
- Equity: Access to essential nutrients is a global justice issue, influencing cognitive development & disease burden
- \text{ATP hydrolysis energy}\approx7.3\,\text{kcal·mol}^{-1}
- 1\,\text{Calorie}=1\,\text{kcal}=1000\,\text{cal}=4184\,\text{J}
- Macronutrient energy densities: \text{CHO}=4\,\text{kcal·g}^{-1},\;\text{Protein}=4\,\text{kcal·g}^{-1},\;\text{Fat}=9\,\text{kcal·g}^{-1}
- Blood glucose homeostasis: 70\text{–}100\,\text{mg·dL}^{-1}\;(3.9\text{–}5.6\,\text{mmol·L}^{-1})
Study Tips & Further Connections
- Cross-link these notes with prior lectures on cellular respiration (glycolysis → TCA → ETC) for mechanistic depth
- Practice drawing metabolic maps to visualise substrate flows & hormonal “switches”
- Apply quantitative skills: calculate caloric requirements, respiratory quotient (\text{RQ}), & Gibbs free-energy changes
- Ethical reflection: evaluate diet fads against biochemical principles above — critical thinking > marketing claims.