Blood Clotting and Disorders
Overview of Blood
Composition: Consists of ~50% blood cells (erythrocytes, leukocytes, platelets) and ~50% plasma.
Platelets (Thrombocytes): Mediate clotting, formed from megakaryocytes in bone marrow. Normal concentration: 150,000-300,000/\mu L. Contain contractile proteins (actin, myosin, thrombosthenin), enzymes for prostaglandins/thromboxane A2 (TXA_2), fibrin-stabilizing factor, PDGF.
Platelet Receptors: Glycoprotein Ib (GPIb) for adhesion; Glycoprotein IIb/IIIa (GPIIb/IIIa) for fibrinogen (aggregation).
Platelet Granules: Dense (\delta) granules (calcium, ATP/ADP, serotonin); Alpha (\alpha) granules (fibrinogen, vWF, plasminogen, PDGF, factors V & VIII).
Plasma: Liquid portion (90% water, 10% solutes), including plasma proteins (immunoglobulins, albumin, apolipoproteins, transferrin, clotting proteins like fibrinogen, prothrombin).
Endothelium: Intact endothelium prevents platelet activation and clotting by:
Smooth surface, glycocalyx (proteoglycans), thrombomodulin (binds thrombin, activates protein C), proPGI2 and NO release, heparin sulfate (activates anti-thrombin III), tissue plasminogen activator (tPA).
Clotting Factors: >50 substances; pro-coagulants (proteins, mostly liver-produced, some require Vitamin K) and anti-coagulants. Balance determines coagulation.
Blood Clotting (Hemostasis)
Hemostasis: Cessation of blood loss from damaged vessels; depends on vessel wall integrity, adequate and functional platelets, adequate and functional clotting factors, and a functioning fibrinolytic pathway.
Stages of Hemostasis:
Primary Hemostasis: Vascular constriction and platelet plug formation.
Vascular Constriction: Due to nervous reflexes, local mediators (TXA2), and decreased vasodilator production (NO, PGI2).
Platelet Plug: Platelets adhere to damaged vessels (via collagen/vWF), release mediators (ADP, TXA_2) to activate and aggregate more platelets, forming a temporary plug.
Secondary Hemostasis (Clot Formation/Coagulation): Blood clotting using intrinsic and extrinsic pathways convergent to a common pathway.
Pathways: Involved intravascular and extravascular elements, platelets, active proteins/factors.
Common Pathway: Prothrombin converted to thrombin; thrombin converts fibrinogen to fibrin monomers; fibrin polymerizes to insoluble meshwork, forming a stable clot (thrombus).
Ca^{++} ions are essential for most steps in the clotting cascade.
Prothrombin: Unstable plasma protein from liver; requires Vitamin K.
Fibrinogen: Large protein from liver; converted to fibrin by thrombin.
Fibrin-stabilizing factor (Factor XIIIa): Strengthens the fibrin meshwork by covalent bonding.
Fibrinolysis (Clot Lysis): Plasminogen (trapped in clot) is converted to plasmin by tPA; plasmin digests fibrin threads and other clotting factors. \alpha_2-antiplasmin inactivates plasmin.
Homeostasis Maintenance: Delicate balance between pro-coagulants (Vitamin K) and anti-coagulants (PGI_2, NO, thrombomodulin, protein C, tPA, antithrombin III, heparin).
Bleeding Disorders
Common Conditions of Impaired Hemostasis:
Vitamin K Deficiency: Leads to insufficient prothrombin, factors VII, IX, X, and protein C, increasing bleeding risk. Causes: malnutrition, malabsorption, antibiotic therapy, biliary obstruction.
Hemophilia: Inherited, X-linked disorders, primarily affecting males.
Hemophilia A: Deficiency of Factor VIII (~85% of cases).
Hemophilia B: Deficiency of Factor IX (\approx 15\% of cases).
Characterized by abnormal bleeding (mild to severe), e.g., hemarthrosis.
Thrombocytopenia: Deficiency in platelet number or function (<150,000/\mu L). Causes bleeding from small vessels, small puncture hemorrhages (thrombocytopenic purpura). Lethal at \% \leq 10,000 counts.
Idiopathic Thrombocytopenic Purpura (ITP): Autoimmune destruction of platelets. Acute (children post-viral), Chronic (adults related to immune disorders).
Thrombocytosis: High platelet counts (>400,000/\mu L). Primary (myeloproliferative disease) or Secondary (stress, exercise, hemorrhage).
Von Willebrand Factor (vWF) Related Disorders: vWF anchors platelets to subendothelium and carries Factor VIII. Deficiency leads to prolonged bleeding from skin/mucosa.
Bernard-Soulier Syndrome: Lack of platelet receptor glycoprotein Ib/IX, impairing adhesion to vWF.
Glanzmann's Thrombasthenia: Deficiency in glycoprotein IIb/IIIa complex, preventing fibrinogen binding and platelet aggregation.
Signs/Symptoms of Bleeding Disorders:
Petechiae: Small, pinpoint red/purple hemorrhages (primary hemostasis defects).
Ecchymosis: Large bruises (>3mm) (secondary hemostasis defects).
Purpura: Purple spots (3-10mm) from bleeding under skin.
Hematoma: Localized blood collection outside vessels.
Hemarthrosis: Bleeding into joint space.
Inappropriate Coagulation (Thromboembolic Conditions):
Disseminated Intravascular Coagulation (DIC): Systemic activation of coagulation leading to widespread microclot formation (thrombosis) and subsequent depletion of clotting factors and platelets, causing secondary hemorrhage (bleeding).
Triggered by trauma, sepsis, malignancy. Can lead to organ failure and circulatory shock.
Thrombus: Abnormal clot forming in a blood vessel.
Embolus: A free-flowing thrombus or other substance (tissue, air, fat, etc.) that can circulate and block vessels (embolism).
Virchow's Triad for thrombus formation: Endothelial injury, sluggish blood flow, increased coagulability.
Bleeding Disorders Caused by Other Diseases:
Vascular Wall Disorders: Fragility due to vessel damage or abnormal formation (e.g., scurvy-Vitamin C deficiency, Cushing's syndrome, geriatric atrophy).
Liver Disease: Impairs synthesis of clotting factors, inhibitors, and affects fibrinolytic system; can also lead to thrombocytopenia and reduced Vitamin K effectiveness.
Medications (Anticoagulants):
Heparin: Increases effectiveness of antithrombin III; rapid effect.
Warfarin: Blocks Vitamin K-dependent synthesis of clotting factors (prothrombin, VII, IX, X).
Antiplatelet Drugs: Inhibit platelet aggregation.
Blood Coagulation Tests
Bleeding Time: Assesses platelet count and function. Normal: 2-8 min.
Clotting Time: Measures clotting process. Normal: 6-10 min.
Prothrombin Time (PT) and International Normalized Ratio (INR): Indicates prothrombin concentration; INR standardizes PT measurements.