AFIB – PVD PHARMACOLOGY Study Notes
AFIB – PVD PHARMACOLOGY
Overview
- Presenter: Penni Merrick, MSN Ed, RN
- Reviewers: E. Hopson, RN, MSN-Ed, CNE & L. Templeton, DNP
Statins: Hyperlipidemia Lowering Agents
Mechanism of Action
- Statin medications decrease cholesterol production in the liver.
- Atorvastatin specifically enhances the number of LDL receptors on hepatic cell surfaces, resulting in decreased LDL levels in the bloodstream.
Medications
- Atorvastatin is a primary example of a statin used in clinical practice.
Client Education
- Patients should alert their medical doctor (MD) if they experience:
- Prolonged muscle aches
- Joint aches
- Muscle tenderness
- Such symptoms may require:
- Holding the medication
- Reducing the dosage
- Switching to another medication
- Patients taking Warfarin should understand that:
- Clotting times may be prolonged while on statin drugs.
- Importance of diet and exercise as adjuncts to pharmacological treatment for hyperlipidemia.
Nursing Implications
- Monitor Liver Function Tests (LFT) and Lipid Panel:
- Baseline assessment followed by re-evaluation at 6 weeks.
- Be aware that rhabdomyolysis has been reported in patients taking atorvastatin.
Anticoagulant Agents
Mechanism of Action
- These agents deplete functional vitamin K reserves, thereby reducing the synthesis of active clotting factors.
Medications
- Warfarin is a commonly prescribed anticoagulant.
Client Education
- Patients should observe for:
- Signs of bleeding that does not stop.
- Eliminate risks for falling, which could exacerbate bleeding.
Nursing Implications
- Monitor for signs of abnormal bleeding, including but not limited to:
- Gastrointestinal (GI) bleeds
- Hematemesis (vomiting blood)
- Intraocular bleeding.
- Regularly check Prothrombin Time (PT) and International Normalized Ratio (INR) levels at least three times a week, aiming for a therapeutic range of [2,3].
Platelet Aggregation Inhibitors
Mechanism of Action
- These medications prevent activation of glycoprotein IIb/IIIa receptors, reducing platelet aggregation (the clumping together of platelets).
Medications
- Clopidogrel is a representative platelet aggregation inhibitor.
Client Education
- Patients should be vigilant about:
- Signs of bleeding that does not stop.
- Risks associated with falling.
Nursing Implications
- Note that there is no reversible agent or antidote for clopidogrel.
- Monitor for abnormal bleeding including:
- GI bleeds
- Hematemesis
- Intraocular bleeding.
- Regularly check Hemoglobin and Hematocrit levels to assess for blood loss.
NSAIDs: Aspirin (ASA)
Mechanism of Action
- Similar to platelet aggregation inhibitors, aspirin prevents activation of glycoprotein IIb/IIIa receptors, thereby reducing platelet aggregation.
Medications
- Aspirin (ASA) is a prominent NSAID used in this capacity.
Client Education
- Patients should monitor for:
- Signs of bleeding that does not stop.
- Gastrointestinal upset, which can escalate to GI bleeding.
- Advise patients with an allergy to ibuprofen that they should not take aspirin.
Nursing Implications
- Monitor for signs of abnormal bleeding, particularly:
- GI bleeds
- Hematemesis
- Intraocular bleeding.
- Be aware that ASA increases the risk of intracranial bleeding.
- Symptoms of mild toxicity from aspirin can include:
- Tinnitus
- Dizziness
- Lethargy
- Nausea
- Vomiting
Low Molecular Weight Heparin (LMWH)
Mechanism of Action
- LMWH works by binding to and potentiating antithrombin III, thereby forming a complex that irreversibly inactivates factor Xa.
Medications
- Enoxaparin is a commonly used LMWH.
Client Education
- Patients should be vigilant for signs of bleeding that does not stop and report:
- Gastrointestinal upset leading to GI bleeding.
Nursing Implications
- Protamine is the antidote for LMWH.
- Ongoing monitoring for abnormal bleeding events such as:
- GI bleeds
- Hematemesis
- Intraocular bleeding.
- Additional observations include:
- Nausea
- Headache
- Confusion
- Injection site irritation or pain.
- Dose adjustments should be made for:
- Advanced age
- Renal insufficiency.
- Typical therapeutic dosing is 1 mg/kg every 12 hours; adjustments are needed for patients older than 75 years.
Activated Factor Xa Inhibitor
Mechanism of Action
- This class of medications prevents the progression of the coagulation cascade through the final common pathway, inhibiting thrombin generation and thereby prolonging clotting times.
Medications
- Rivaroxaban represents this category of anticoagulant.
Client Education
- Patients should be aware of:
- Signs of bleeding that does not stop.
- Gastrointestinal upset leading to GI bleeding.
- Monitoring of liver enzymes is necessary.
Nursing Implications
- Andexanet alfa serves as the antidote for rivaroxaban.
- Monitoring for abnormal bleeding signs:
- GI bleeds
- Hematemesis
- Intraocular bleeding.
- Before initiating treatment, patients should undergo a screening for:
- Bleeding disorders
- Coagulation profiles
- Hepatic or renal impairments.
- Routine coagulation testing is not necessary for patients on rivaroxaban.