Cannabiniods (weed)
Cannabis’s role in society
long his of use often medical
Historically, marijuana was replaced by more effective drugs in the medical fields and then outlawed
Research opened up cannabis use for new med appilcations and legalizations
research
very very hard to get acesses to research
needs a lot of approval from fed gov
doesn’t matter if the state it is makes it legal, it is still very heavily montored in studies
lots of legal loopholes
there are more compunds in plant matter than just a single agonist effecting 1 transmiter
Cannabioids as a drug class
Major active ingredent: ^9- tetrahyrocannabinol (THC)
when smoked, produces a mix of hallucinogentic, depresant, and stimulant effects, known as cannabis intoxication
Targets the CB receptors (retro messengers)
Most of the effects last 2-6hrs
Other forms of THC
Delta 8 THC
THCA
these get converted into THC when heated
Synthetic THC
Leagal loop holes
Cannabidiol
No high
Potential med benifits
Forms
Natural forms
Produced from varties of hemp plants
Hash: Solidified resin of the cannibis plant
Marijuana: mix of bud, crushed leaves, and flowering tops
Extracts/concentrates: THC extracted and suspended in a medium (vape pen)
Edibles/ tinctures: THC is bound to a fat and ethier cooked or applied to skin
Potency varies, edibles may be a black box of potency, this matters for user experance, edibles can take 2-4 hours to kick in and may take a long time to wear off (go low on edibles)
Synthetic forms
“K2” or spice- often sold as incense at gas stations
black market versions- quality control is an issue here
(NOT SAFE)
Medical use of THC
pain mangement (CB1/CB2 agonists)
transdermal apllication might be esspiaclly effective
more work on the CB1 than CB2 receptors
Changes to hunger circutry
weight loss prevention- eating disorder/cancer
nausa control- kemo threapy
Movement control
Pakingsons- helps with, relives symptoms, helps with circuts in basial ganglia and it changes the firing and helps smooth out movements
seizures
Glaucoma :)
pressure in the eyes
CBD and med benifits
Anxiety: studies/clinic trials are exploring the common report that CBD can reduce anxiety
insomina: studies suggest that
chronic pain
addiction
Cannabis use disorder
Influanced by reg use
social and occupational lives of 1.6% of people in US are effected, including high # of highschool/college
The lifetime risk of reg cannabis users becoming dependent on cannabis is 9%
the current varieties of marijuana are 7 times more powerful than those found in 1970’s due to higher THC content (15%)
Edibles and concentrates are also highly potent
Dangers
tolerance and withdrawl sysmptoms
occasional panic reactions, automible accdents, and decreased mem while high
Long term health prob, reprofuction issues
psychosis and mental health issues
Tolernace
tolernace does build
it seems to primarally be a change in the receptor dynamics and availbitlity in the synapse
Role in addiction circut
Cannabinioids increase dopamine
also increase endogenous (natural) opioid relase (so the role opioids in addiction is also part of story here too)
Cannabiniods as a retro messenger affect glutamate excitation in the VTA
Role in VTA
retro messengers reduce firing rate
Can sepress excitation
if glutamate neurons that excite the VTA are hit they will reduce their excitation
Can increase exciation
I
Impact on necleus accumbens
it depends
may be why THC has less addcitive tendancys
reasleases dopamine randomly, sometimes increases dopamine sometimes inhinits dopamine,
depends whats going on in brain when it hits (mental state and neural circutry)
wi
Withdrawl
many of the withdrawl sysmptoms are offten the opp of the effect of drug
Insomina
aneroxia
anxiety
irrablitity
depresion tremors
Does and durration effect severity of withdrawl