Introduction to Quality Control

PHARMACEUTICAL ANALYSIS 2

(Instrumental Methods of Analysis)

TOPIC 1: INTRODUCTION TO

QUALITY CONTROL

2nd Semester, SY 2023 - 2024 PRELIM - Pharmaceutical Analysis 2 (PHAN212)

Learning Outcomes:

At the end of this unit, the students are expected to:

Define and discuss pharmaceutical analysis and its importance

in the pharmaceutical industry.

Recognize the ICH Quality guidelines.

Differentiate the different types of errors in analysis.

Differentiate accuracy from precision.

Discuss the validation of analytical procedure.

Define quality control, quality assurance and other related

terms.

Describe the quality control organizational chart and the QC

system.

Differentiate the QC divisions by their functions.

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

Unit Outline:

• Pharmaceutical Analysis

• Errors in analysis

• Accuracy and Precision

• Validation of analytical procedure

• Introduction to quality control

• Quality Control System

• Total Quality Management

• Accreditation (ISO)

• Organization of Quality Control

• Common divisions in a manufacturing firm

• Control functions

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

Checklist

Attend Onsite Lecture

Duration: 3 hours

Read course and unit outcomes.

Read study guide prior to onsite

attendance.

Read required learning resources.

Proactively participate in onsite

discussions.

Answer and submit course unit

tasks.

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

The development of the

pharmaceuticals brought a revolution

in human health.

These pharmaceuticals

would serve their intent only

if they are free from

impurities and are

administered in an

appropriate amount.

SOURCE: Masoom Raza Siddiqui, Zeid A. AlOthman, Nafisur Rahman, Analytical techniques in pharmaceutical analysis: A review , Arabian Journal of Chemistry, Volume 10, Supplement 1, 2017, Pages S1409 - S1421,

ISSN 1878 - 5352,

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

To make drugs serve their purpose, various chemical and

instrumental methods were developed at regular intervals

which are involved in the estimation of drugs.

SOURCE: Masoom Raza Siddiqui, Zeid A. AlOthman, Nafisur Rahman, Analytical techniques in pharmaceutical analysis: A review , Arabian Journal of Chemistry, Volume 10, Supplement 1, 2017, Pages S1409 - S1421,

ISSN 1878 - 5352,

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

These pharmaceuticals may develop impurities at various stages of

their development, transportation and storage which makes the

pharmaceutical risky to be administered thus they must be

detected and quantitated.

SOURCE: Masoom Raza Siddiqui, Zeid A. AlOthman, Nafisur Rahman, Analytical techniques in pharmaceutical analysis: A review , Arabian Journal of Chemistry, Volume 10, Supplement 1, 2017, Pages S1409 - S1421,

ISSN 1878 - 5352,

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

For this, analytical instrumentation

and methods play an important

role.

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

What is

Pharmaceutical

Analysis ?

• It is a branch of practical chemistry that

involves a series of process for

identification, determination,

quantification and purification of a

substance, separation of the

components of a solution or mixture, or

determination of structure of chemical

compounds .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

SOURCE: Watson, David G., Pharmaceutical Analysis: A Textbook for Pharmacy Students & Pharmaceutical Chemist, 4th ed. 2017. Elsevier. ISBN: 978 - 0 - 7020 - 7029 - 7

Pg. 2

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

International

Conference on

Harmonisation (ICH)

• International Conference on Harmonisation of Technical

Requirements For Registration of Pharmaceuticals for

Human Use

• Addressed the requirements for control of the quality of

methods of analysis ( validation ) .

• Initiated in Brussels in 1990

• Representatives of regulatory agencies and industry

associations of Europe, Japan and the USA .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

International

Conference on

Harmonisation (ICH)

PURPOSE : to standardise the requirements for medicines

regulation throughout the world .

Most important analytical procedures that require validation are:

• Identification tests

• Quantitative tests for impurities

• Limit tests for the control of impurities

• Quantitative tests of the active moiety in samples of drug

substance or drug product or other selected component(s) in the

drug product.

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

With such large amounts of money being spent on

analytical quality control, great importance must be

placed on providing accurate and precise analyses.

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

2 TYPES OF CHEMICAL ANALYSIS

Quantitative

Qualitative analysis analysis

• is performed to establish • techniques are mainly used to

composition of natural/synthetic quantify any compound or

substances . substance in the sample .

Examples : Examples :

• Distillation, extraction, color • Titration, gravimetric analysis,

change, chromatography, etc . etc .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

TYPES OF ERRORS

ERROR

- may be defined as a deviation from the absolute value or

from the true average of a large number of results .

1 ) Determinate or constant 2 ) Indeterminate errors

- are those that, although - caused by uncontrollable

sometimes unsuspected, may be fluctuations in variables that

avoided or determined and affect experimental results

corrected once they are

uncovered .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

ERRORS IN ANALYSIS

1 . Gross Error

- takes into account human oversight and other mistakes

while reading, recording, and readings .

- easily recognized since they involve a major breakdown in

the analytical process such as :

• samples being spilt,

• wrong dilutions being prepared or

• instruments breaking down or being used in the wrong way .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

ERRORS IN ANALYSIS

2 . Random Error

- the random errors are those errors, which occur irregularly

and hence are random .

- these can arise due to random and unpredictable

fluctuations in experimental conditions

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

ERRORS IN ANALYSIS

3 . Systematic Error

- ENVIRONMENTAL 🡪 arises in the measurement due to the effect of

the external conditions on the measurement .

• Examples : temperature, pressure, humidity

- OBSERVATIONAL 🡪 arise due to an individual’s bias, lack of proper

setting of the apparatus, or an individual’s carelessness in taking

observations .

- INSTRUMENTAL 🡪 arise due to faulty construction and calibration of

the measuring instruments .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

ACCURACY and PRECISION

In an experiment, PRECISION is

defined as the reproducibility of

results and measurements,

while ACCURACY refers to how

close the value is to the actual or

true value .

It may be that the results are both

accurate and precise, neither or

accurate but not precise or not

accurate but precise .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

ACCURACY and PRECISION

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

SOURCE: Watson, David G., Pharmaceutical Analysis: A Textbook for Pharmacy Students & Pharmaceutical Chemist, 4th ed. 2017. Elsevier. ISBN: 978 - 0 - 7020 - 7029 - 7

Pg. 5

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

VALIDATION OF ANALYTICAL

PROCEDURE

The Analytical Procedure

- provides an exact description of how the analysis is carried out.

- It should describe in detail the steps necessary to perform each analytical test.

The full method should describe:

i. the quality and source of the reference standard for the

compound being analyzed

ii. the procedures used for preparing solutions of the reference

standard

iii. the quality of any reagents or solvents used in the assay and their

method of preparation

iv. the procedures and settings used for the operation of any

equipment required in the assay

v. the methodology used for calibration of the assay and

methodology used for the processing of the sample prior to

analysis.

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

“ QUALITY ”

• is the combination of attributes or

characteristics of a product which, when

compared to a standard, serves as a basis

for measuring the uniformity of the product

and determines its degree of acceptability .

“ CONTROL

• Refers to the measure or step that is used to

prevent or eliminate drugs risks /hazards to

make it safe & effective .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

QUALITY CONTROL

• Is a tool, which gives the assurance

that a product conforms to standards

and specifications through the system

of inspection, analysis and action .

• The operational techniques and

activities used to fulfill requirements

for quality,

• To assure safe, pure and effective

drug product .

• Quality is everybody’s business .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

QUALITY ASSURANCE

• The sum total of the organized

activities performed with the

intent to ensure that all active

pharmaceutical ingredients are of

the quality required for their

intended use .

• All the planned and systematic

activities implemented in a quality

system so that quality

requirements for a product or

service will be fulfilled (American

Society for Quality, ASQ) .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

QA QC

Set of preventive Detection activities

activities

Ensures that standards are Defines the standards to be

followed at every step followed

Process - oriented Product - oriented

Focus on defect Focus on defect

prevention identification

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

QUALITY

CONTROL

SYSTEM

- established at the conception of a

new product, during production of

the batch, and during distribution of

the commercial package .

- This system is a combination of

those administrative and technical

procedures, which must be used to

produce and deliver a safe, pure,

and effective product to the end

user .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

QUALITY

CONTROL

SYSTEM

Guarantees that the drug product is :

Free from impurities

Physically and chemically stable .

Having the amount of active ingredient as stated on the

label .

Providing an optimal release of active ingredients when

the drug product is administered .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

QUALITY

CONTROL

SYSTEM

BENEFITS :

1 . The system minimizes or eliminates the risk of

marketing unsafe products

2 . It guarantees conformance to regulatory

requirements

3 . It guarantees product efficacy

4 . It reduces operating costs

5 . It reduces operating losses

6 . It produces higher employee morale

7 . It motivates the pharmaceutical/medical professions

to sell or prescribe the product

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

• a process inside an organization with the aim to improve

its performance by learning about good practices for

primary and/or support processes through looking at

those processes in other, better - performing

organizations, building on evaluation of relevant

performances in own and other organizations .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

TOTAL QUALITY

MANAGEMENT (TQM)

• A management approach for an

organization, centered on quality,

based on the participation of all

its members and aiming at long -

term success through customer

satisfaction, and benefits to all

members of the organization and

to society .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

Primary

Elements of

Total Quality

Management

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

ACCREDITATION

• Quality assessment with an

attached judgment that the

evaluated unit (program or

organization) is good enough to

have the right to exist in a

particular system .

• Often, accreditation is given for a

limited period of time (usually

between 4 and 10 years) and is

repeated in a cyclical process at

the end of the period of validity .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

• Popular name for International Organization For

Standardization .

• A voluntary, non - treaty federation of standards setting bodies

of some 130 countries . Founded in 1946 - 47 in Geneva as a UN

agency, it promotes development of standardization and

related activities to facilitate international trade in goods and

services, and cooperation on economic, intellectual, scientific,

and technological aspects

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

ORGANIZATION OF QUALITY

CONTROL

Part of a manufacturing firm is a defined

organization .

⮚ functions and responsibilities

⮚ effective coordination

⮚ all activities are performed towards the production

of a product of the highest standard and at the

lowest cost .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

COMMON DIVISIONS IN A

MANUFACTURING FIRM:

1. Finance

2. Production

3. Quality Assurance (Quality Control)

4. Marketing (optional in a third - party contract

manufacturer)

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

CONTROL FUNCTIONS:

Control functions may appear varied and never quite

identical in any two companies by basically, these

functions can be classified into four categories :

1. Analysis Function

2. Monitor Function

3. Record Review and Release Function

4. Audit Function.

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

1. Analysis Function

⮚ To assure the acceptability of a product .

⮚ Conducts testing on the raw materials and packaging

components and bulk products :

during processing

after packaging

after distribution

⮚ Product against which a complaint is registered may also be

analyzed to determine its validity and the cause of the reported

deficiency .

⮚ Appropriate steps may then be taken to prevent recurrence of

similar problem .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

2. Monitor Function

⮚ To sample and examine materials

⮚ To assure that even though production personnel have the

primary responsibility for control over their processes, these

processes are maintained and that any deviation from specified

requirements is reported .

⮚ To conduct environmental monitoring .

⮚ To control the microbial and particulate matter content of

environmental air in areas where pharmaceuticals such as

parenterals are processed .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

3. Record Review and

Release Function

⮚ To determine accuracy and

completeness of all records

generated during the course of

production prior to the release

of each lot of finished product

to the market .

⮚ A detailed checklist is

frequently employed by the

reviewer .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

4. Audit Function

⮚ To train employees to comply with

the SOP’s and to understand why

and how these SOPs are to be

followed .

⮚ The quality audit is designed to

detect areas where the established

SOPs are not being followed and to

report these findings to the

supervisor for appropriate action .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

QUALITY CONTROL

DIVISIONS

A. Materials Inspection Section

B. Analytical Laboratory

C. Biological Testing Laboratory

D. Quality Coordination Office

E. Specification and Analytical

Development

Figure 1: shows a typical organization within the quality control department.

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

A. Materials Inspection Section

Inspectors are alert individuals

who had experience and who are

familiar with the physical

characteristics of the materials they

sample and are well versed in

sampling techniques .

Inspection stations are placed in the area of operation,

warehouse, manufacturing and packaging areas .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

A. Materials Inspection Section

The functions of this section are:

1. To sample and examine all raw materials received.

2. To sample and conduct physical tests on:

• All shipments of packaging materials

• All manufacturing, filling and packaging operations

3. To maintain periodic examination on the quality of

inventories throughout all phases of storage, shipping

and distribution .

4. To perform an audit which is independent of the

work done byproduction personnel

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

B. Analytical Laboratory

• The analytical laboratory should be in an

accessible area and protected from noise and

vibration common to manufacturing

operations .

• This division performs all qualitative and

quantitative analysis on raw materials,

intermediate and finished products .

⮚ The analysts should know the usual gravimetric and

volumetric analysis .

⮚ They should be skillful in handling instruments

(Spectrometry, Aqueous and Non - aqueous titrimetry,

Chromatography)

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

C. Biological Testing

Laboratory

⮚ The staff in a biological testing laboratory should be well

trained and experienced in both simple and complex

microbiological procedures and biological interactions .

⮚ A veterinarian is recommended to supervise the care and

maintenance of the various species of animals used in the

tests .

⮚ The area :

should be provided with particular rooms where

biological tests are conducted .

should be protected against noise specifically the

areas where animals are used .

should be provided with an animal house so maintained

and is a separate unit from the main laboratory, if

necessary .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

C. Biological Testing

Laboratory

⮚ The staff in a biological testing laboratory should be well

trained and experienced in both simple and complex

microbiological procedures and biological interactions .

⮚ A veterinarian is recommended to supervise the care and

maintenance of the various species of animals used in the

tests .

⮚ The area :

should be provided with particular rooms where

biological tests are conducted .

should be protected against noise specifically the

areas where animals are used .

should be provided with an animal house so maintained

and is a separate unit from the main laboratory, if

necessary .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

C. Biological Testing

Laboratory

The functions of this division are :

1. To perform and evaluate

microbiological and pharmacological

assays, sterility, pyrogen and

bacteriological tests, irritation, safety

or acute toxicity tests .

2 . To conduct environmental monitoring .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

D. Specification and Analytical

Development

This section should have firm background not only in the

principles of quality control and analytical procedures but also in

manufacturing, research, product development and in statistics in

order to perform the following functions :

1. To coordinate with research, product development,

production, sales and management towards improvement

of a product.

1. To establish specifications for raw and packaging materials.

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

D. Specification and Analytical

Development

Other functions of this division are :

3 . To validate existing and tentative

procedures of testing .

4 . To establish specifications based on

validated procedures .

5 . To develop new assay methods for in -

house use .

6 . To develop and improve

specifications for quality characteristics

of the final product being manufactured .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

E. Quality Coordination Office

⮚ This section should be accessible to all

manufacturing and packaging operations

since documentation is its main

responsibility .

⮚ The functions of this section are :

1. To maintain and store records that represent

the history of the batch from start to finish .

These records include the batch and master

formula records, raw material analytical

records, printed and packaging material

inspection reports and retention files .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

E. Quality Coordination Office

Other functions of this division are:

2 . To be able to furnish data that will aid in analyzing product performance

in the market . These documents are the stability studies and returned

goods reports .

3 . To investigate customer complaints or inquiries on product quality and

to forward the results of the investigations in the form of technical

reports to the sales organization .

4 . To call the attention of the appropriate development group any aspect

that provides a basis for improvement of a product for consideration and

action .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

E. Quality Coordination Office

Other functions of this division are:

5 . To provide data that give scientific and legal status, i . e . , data

generated from the use of recognized standard compendia . This

is essentially a function of the distribution section or warehouse .

6 . To maintain and develop SOP’s .

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

OTHER AREAS IN MANUFACTURING

FIRM THAT A PHARMACIST CAN WORK:

Marketing

Medical Affairs

Medical Liaisons

Research and Development

Production

Legal or Regulatory Affairs

Administration

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

1. Define cGMP

2. Define and explain quality control in pharmacy.

3. Differentiate QA from QC

4. What is the importance of quality in pharmaceutical

products?

5. Define TQM.

6. What are the control functions in quality control?

7. Enumerate the benefits of QCS.

8. What is the importance of accreditation in an institution?

9. What is an SOP? Give its importance in manufacturing

procedures.

10. TRUE OR FALSE. Inspection stations are placed in the

area of operation, warehouse, manufacturing and

packaging areas.

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

Watch this video:

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oYXJtYWNldXRpY2FsIGluZHVzdHJ5

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

References:

Jenkins, Glenn L, Jenkins Quantitative Pharmaceutical

Chemistry, N . Y, N . Y . : Mc Graw, Latest Edition

Watson, David G . , Pharmaceutical Analysis : A

Textbook for Pharmacy Students & Pharmaceutical

Chemist, 4 th ed . 2017 . Elsevier . ISBN : 978 - 0 - 7020 -

7029 - 7

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

Activities for next meeting:

1 . Quiz No . 1 : Introduction to Quality Control

2 . Assignment No . 1 : Quality Control

3 . Lecture Topic : Quality Control

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)

THANK YOU!

Any questions?

You can find me at:

username@fatima.edu.ph

2nd Semester, SY 2023 - 2024 PRELIM - Pharmaceutical Analysis 2 (PHAN212)

OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)
ERRORS IN ANALYSIS
2. Random Error
- the random errors are those errors, which occur irregularly
and hence are random.
- these can arise due to random and unpredictable
fluctuations in experimental conditions






OLFU - College of Pharmacy PRELIM - Pharmaceutical Analysis 2 (PHAN212)
ERRORS IN ANALYSIS
3. Systematic Error
- ENVIRONMENTAL 🡪 arises in the measurement due to the effect of
the external conditions on the measurement.
• Examples: temperature, pressure, humidity
- OBSERVATIONAL 🡪 arise due to an individual’s bias, lack of proper
setting of the apparatus, or an individual’s carelessness in taking
observations.
- INSTRUMENTAL 🡪 arise due to faulty construction and calibration of
the measuring instruments.





ACCURACY and PRECISION
In an experiment, PRECISION is
defined as the reproducibility of
results and measurements,
while ACCURACY refers to how
close the value is to the actual or
true value.
It may be that the results are both
accurate and precise, neither or
accurate but not precise or not
accurate but precise.