HIV
Discuss the epidemiology of HIV
Identify sources of HIV transmission and methods for prevention
Identify patients who should be screen for HIV
Describe the HIV life cycle and identify current targets of antiretroviral therapy
Describe the pathogenesis, diagnosis, and course of HIV infection
Identify complications associated with HIV including opportunistic infections
Identify candidates for antiretroviral therapy and opportunistic infection chemoprophylaxis
What is the first ARV that was FDA approved?
Zidovudine (AZT)
What population was 2/3 of new HIV diagnoses in 2022?
Black and Hispanic people
Although HIV transmission has gone down, what age group has an increasing incidence rate?
25-34 and 35-44
Although HIV transmission has gone down, what race/ethnic groups has an increasing incidence rate?
American Indian/Alaska Native, Hisptanic/Latino and Native Hawaiiain and other Pacific Islander
What treatment should all HIV infected patient receive?
Antiretroviral Therapy (ART)
What is Antiretroviral Therapy used for?
Reduce morbidity & mortality and prevent transmission of HIV
When should patients infected with HIV start on ART?
immediately after HIV diagnosis to increase the uptake of ART and linkage to care, decrease viral suppression time for individual patients, and improve virologic suppression rate
What 4 studies combine results found zero HIV transmission where the HIV infected partner had durable suppression.
HPTN-052, Opposites Attract, Partners 1 & 2
List the HIV care continuum
Diagnosed with HIV → Linked to Care → Receipt to Care → Retained in Care → Viral Suppression
What is PreExposure Prophylaxis (PrEP)?
Antiretroviral therapy that’s given to prevent infection before potential exposure
What is Post Exposure Prophylaxis (PEP)
Antiretroviral therapy that’s given within 72 hours of exposure to reduce the risk of infection
Describe the regimen required for PEP
3 ARVs daily for 28 days
What are the 3 main transmission routes
Sexual, Parenteral, Mother-to-Child
Describe how sexual contact is a vehicle for transmission.
Blood, Semen, and Vaginal Secretion
Describe how parenteral is a vehicle for transmission.
Sharing needles/syringes, Infected blood transfusion products, Accidental contact of sharp object trauma
Describe how mother to child is a vehicle for transmission.
Vertical transmission and Breastfeeding
What transmission route is the most common?
sexual contact
What are factors that increase the risk of transmission for sexual contact?
Concurrent STDs (ulcerative lesions), More infectious partner (higher viral load), Lack of male circumcision, Vaginal bleeding
What are preventative measures for sexual contact transmission?
Abstinence, Monogamy, Barrier precautions, Reduction of high-risk behaviors, ART, PrEP, PEP
What are factors that increase the risk of Parenteral transmission?
Exposure to contaminated blood, Intravenous Drug Use (IVDU) (used/contaminated needles), Blood transfusions, Transplanted organs, Mucocutaneous exposure (eyes, mouth, nose), Percutaneous needle stick
What are preventative measures for parenteral transmission?
substance use treatment programs, needle exchange programs, sterilization of drug paraphernalia, PrEP, Receipt of contaminated blood products
What are factors that increase the risk of mother-to-child transmission?
during/near time of birth, prolonged rupture of membranes, genital infection during pregnancy, preterm delivery, vaginal delivery, birth weight < 2500 gm, illicit drug use during pregnancy, HIV maternal viral load
According to USPSTF, what population should be recommended to be screened for HIV?
15-65, those outside the range with an increased risk, and all pregnant persons
How often of those with known risk be screened?
annually
Explain the HIV life cycle between days 0-2.
Exposure to HIV, Virus collected by dendritic cells and carried to lymph nodes
Explain the HIV life cycle on day 3
HIV replicates in CD4 cells, released into blood, and spread to other organs
Explain HIV life cycle after day 3
Continued viral replication → massive CD4 T-cell destruction → viral spread to multiple organs (brain, spleen, regional & distal lymph nodes, bone marrow)
What are the targets of HIV infection and why?
CD4 T Helper Lymphocytes (TH1, TH2, TH17) activate macrophages, stimulate B-cell made Abs, recruit neutrophils for infection sites, regulate and limit immune response to prevent autoimmune responses
Describe the HIV virus components
Capsid
HIV’s core that contains HIV RNA
Envelop
Outer surface
Enzymes
Proteins that carry out steps in HIV life cycle
Glycoproteins
Protein spikes embedded in the Envelope which attach and fuse with CD4 cells
RNA
Genetic material
List the steps of the HIV life cycle
Binding/Attachment
Fusion
Reverse Transcription
Integration
Replication
Assembly
Budding
Explain Step 1: Binding
HIV binds to CD4+ → binds to co-receptor
What HIV therapy drugs are seen targeting in the binding step?
Enfuvirtide, Fostemsavir, Ibalizumab, Maraviroc
Explain Step 2: Fusion
after binding to the co-receptor the HIV envelope fuses with the CD4 cell membrane → spills viral contents into the cell (HIV RNA and Viral Enzymes — Reverse Transcriptase, Integrase, and Protease)
Explain Step 3: Reverse Transcription of HIV RNA
Reverse Transcriptase converts HIV RNA → HIV DNA which enters the CD4 nucleus and combine with cellular DNA
What HIV therapy drugs target Step 3 of Reverse Transcriptase
Nucleoside Reverse Transcriptase Inhibitors (NRTIs)
Tenofovir, Abacavir, Emtricitabine, Lamivudine
Non-Nucleoside Reverse Transcriptase Inhibitors (NNRTIs)
Rilpivirine, Doravirine, Efavirenz
Explain Step 4: Integration of Viral DNA into Host DNA
Integrase joins viral and host DNA
What HIV therapy drugs target (Integrase inhibitors) Step 4 of Integration
Dolutegravir, Bictegravir, Raltegravir, Elvitegravir, Cabotegravir
Explain Step 5: Replication
Host begins to create long chains of HIV proteins which are building blocks for more HIV viruses
Explain Step 6: Assembly
New HIV RNA and HIV proteins made by the host CD4 cell move to the cell surface a d assemble into immature (noninfectious) HIV
Explain Step 7: Budding
Immature HIV virus pushed out from host CD4 cell and the long protein chains is cleaved by viral Protease
Protein chains form new functional HIV proteins → mature virus
What HIV therapy drugs (Protease inhibitors) target Step 7 for budding?
Darunavir
Atazanavir
Explain the typical course of HIV infection
after initial infection (acute HIV syndrome) → spiked viral load with a drop in CD4 count
after some weeks, CD4 begin to recover and the body starts to build immunity → drop in viral load (clinical latency period — can be years)
rise in viral load and sinking CD4 count until progression to AIDs or immunodeficiency syndrome
What is Acute HIV Syndrome?
when HIV enters the body and infects a large number of CD4+ cells
due to high viral load, patients are high risk of transmitting
What symptoms are seen during Acute HIV Syndrome?
Flu-like symptoms
Fevers, Chills, Rash, Night Sweats, Sore Throat, Fatigue, Swollen Lymph Nodes, Mouth Ulcers
When do symptoms begin for Acute HIV Syndrome?
1-4 weeks pose exposure and lasts ~2-4 weeks
Explain the Clinical Latency period in Acute HIV Syndrome
begins 2-4 weeks after exposure
viral load falls to a set point
CD4 cells rebound
viral replication is ongoing and CD4 count will steadily decrease
Explain the period that lead the Progression to AIDs
immune system deteriorates
viral load increases while CD4 count drops to dangerously low levels
patient at risk to develop various Opportunistic Infections (OIs)
What is the median time period of typical progressors (90%)
7-12 years
What is the median time period of rapid progressors (<10%)
< 3 years
What is the median time period of long term non-progressors (<1%)
> 15 years
normal, stable CD4 count and viral load of < 500 copies/mL
Explain why CD4 count are markers of disease progression
normal: 500-1600
assess immunologic response to therapy
determines when to initiate chemoprophylaxis for OIs
entry into care, 3-4 months after ART initiation or change in drug therapy and periodically thereafter
Explain why HIV viral load are markers of disease progression
# of HIV RNA copies per mL of plasma
each viral load test has a lower limit of detection
assess virologic response to therapy
entry into care, 2-8 months after ART initiation or change in drug therapy and every 3-4 months thereafter
viral load should decrease 1 log in 2-8 weeks after initiating therapy
Explain the criteria for AIDs diagnosis
CD4 < 200 cells/mm3
presence of OI or AIDs defining illness
Oropharyngeal candidiasis
Cryptococcus
Pneumocystis pneumonia
Toxoplasmosis
Recurrent bacterial pneumonia
Mycobacterium avium complex
Kaposi’s sarcoma, other AIDs defining malignancy
HIV associated wasting syndrome
What OI is likely to infect a patient with a CD4 cell count ~200
Oropharyngeal candidiasis and Pneumocystis pneumonia
What OI is likely to infect a patient with a CD4 cell count ~100
Toxoplasmosis encephalitis and Cryptococcus meningitis
What OI is likely to infect a patient with a CD4 cell count ~50
Mycobacterium avium complex and Cytomegalovirus retinitis
What are the diagnostic tests for HIV
Antibody test (EIA)
detects HIV Abs
Rapid HIV screens
~23-90 days after exposure
Antigen/Antibody Test
most common in labs
~18-45 days after exposure
Nucleic Acid test
viral load testing
~10 days after exposure