Chapter 24
Chapter 24: Glycogen Degradation Overview
Focuses on:
Glycogen-degrading enzymes.
Regulation of glycogen phosphorylase.
Role of intercellular signaling in glycogen breakdown.
Key Concepts in Glycogen Degradation
Glycogen synthesis and degradation are co-regulated with glycolysis and gluconeogenesis (see Chapters 16 and 17).
Glycogen Structure
Glycogen is a polymer of glucose, functioning as an energy storage molecule in animal cells.
Rapid mobilization of glucose for energy occurs mainly in the absence of oxygen, supporting brain and red blood cells.
Structure features:
Glycogen granule nucleated by glycogenin (dimeric protein).
Branches occur approximately every twelve residues.
Muscles contain about 2% glycogen by weight (for movement) while the liver harbors around 10% (for sustaining blood-glucose levels).
Major reactions occur at non-reducing ends of glucose chains.
Glycogen Degradation Enzymes
Glycogen Phosphorylase: Key enzyme that cleaves glycogen chains.
Converts glycogen into glucose 1-phosphate through phosphorolysis rather than hydrolysis, requiring Pi.
Phosphate addition activates the product, preventing ATP usage and retaining glucose within the cell.
Additional Enzymes Needed for Branch Points:
Transferase: Moves glucose residues from one branch to another.
α-1,6-Glucosidase (Debranching Enzyme): Hydrolyzes 1,6 linkages, allowing full glucose extraction.
Hexokinase: Phosphorylates released glucose from debranching.
Phosphoglucomutase: Converts glucose 1-phosphate to glucose 6-phosphate for glycolytic entry.
Disease Associated with Glycogen Breakdown
Failures in debranching enzymes can lead to genetic diseases.
Hers Disease: A hereditary disorder due to mutations in the liver isozyme of glycogen phosphorylase, causing liver enlargement and low blood glucose levels.
Regulation of Glycogen Phosphorylase
Types of Phosphorylase:
Phosphorylase a: Active, phosphorylated form.
Phosphorylase b: Inactive, non-phosphorylated form.
Conformation states:
R State (Relaxed): More active.
T State (Tense): Less active and partially blocked.
Tissue-Specific Regulation:
Muscle: B form predominant at rest, activated during exercise.
Liver: A form is typically active, modulated by glucose levels.
Allosteric Regulation in Muscle and Liver
Muscle:
Energy charge modulates activity: High ATP/Glucose 6-Phosphate stabilizes T state (inhibitory).
Low ATP/High AMP activates phosphorylase (R state).
Liver:
Active unless free glucose is present.
Hormonal control via insulin (dephosphorylation) and glucagon (phosphorylation).
Hormonal Regulation
Epinephrine: Stimulates glycogen breakdown in muscles and liver during activity.
Glucagon: Signals low glucose levels, promotes breakdown in the liver.
Both hormones regulate phosphorylase via G-protein linked signaling pathways.
Summary of Key Enzymatic Activities in Glycogen Degradation
Six crucial enzymes:
Glycogen Phosphorylase: Initial cleavage.
Transferase: Moves branches.
Debranching Enzyme: Completes degradation.
Hexokinase: Phosphorylates glucose.
Phosphoglucomutase: Converts glucose 1-P to glucose 6-P.
Glucose 6-Phosphatase: Exclusively in the liver for glucose export.
Key Concept Questions
Glycogen structure, glycosidic bonds, and enzymatic actions involved in degradation are essential for understanding glucose metabolism.