The Dosage Form

To correctly process a written medication order, it is necessary to know some

basic terminology. When the drug is prescribed, it is usually prescribed in

a specifi c dosage form. The form in which the drug is used depends on

the condition of the patient. Most drugs are taken in tablet form orally (by

mouth), but others must be used in a suppository form (e.g., for a vomiting

patient), topically, in the eye, systemically, on the skin (for a rash or

skin condition), or in oral liquid form (for a child). Some drugs may also be

administered through the skin, via the transdermal patch.

Since different dosage forms are packaged and used differently, it is important

to know which dosage form the drug must be in. In addition, the instructions

written by the prescriber on the prescription form are abbreviated, and

the technician must be familiar with these abbreviations to accurately convey

the instructions to the patient. (See Table 2-1 and Appendix B.)

Solid Dosage Forms

Solid dosage forms are those that can be picked up and handled. These include

the oral dosage forms of tablet, capsule, and enteric-coated tablet

(Figure 2-1).

The Tablet

A tablet is made of pressed powder. How hard the powder is pressed determines

how the tablet can be used. For example, a sublingual tablet is made

to dissolve quickly, under the tongue, and therefore cannot be pressed hard

into a dense tablet. (Since the tablet is so soft, it must be handled very carefully

to avoid turning it into a pile of powder.) An example of a sublingual

tablet would be a nitroglycerin tablet, which is made to dissolve quickly so

that the drug may be rapidly absorbed into the system.

Most tablets are lightly coated with a protective coating (a “fi lm” coating)

to protect the drug. This is does not affect the absorption or dissolution of

the medication. An enteric tablet is coated with a hard-shell coating, designed

to protect the drug from acid in the stomach. The drugs contained in enteric

tablets are normally best absorbed in the basic pH of the duodenum. An

exception is enteric-coated aspirin, which is coated so that it will not dissolve

in the stomach and subject the stomach lining to its effects. Enteric-coated

tablets should not be split or crushed.

The Capsule

A capsule is a gelatin “container” fi lled with powdered drug, drug granules,

a liquid drug formulation, or an oil. Examples would be antibiotics capsules,

liquid vitamins (e.g., A, D, or E), and many over-the-counter cold remedies.

Other Solid Dosage Forms

Other dosage forms, which are less frequently prescribed and solid in nature,

include:

• The lozenge: a hard tablet or molded shape containing drug in a sweetened,

fl avored base. The lozenge is designed to be held in the mouth

while it slowly releases drug for oral absorption. This dosage form is

particularly useful for administration of pain medication for chronic pain

and for the relief of nausea during cancer chemotherapy. Drugs available

in lozenge form are listed in Table 2-2.

• Drug powders for inhalation: In this dosage form, a very fi ne crystalline

form of the drug (a microcrystalline powder) is mixed with an inert sugar

(e.g., lactose) and packaged into a single-dose “blister.” The blister is then

inserted into a special apparatus called a “diskhaler,” which pierces the blister,

aerosolizes the drug, and allows the patient to inhale the medication.

Table 2-2 Drugs Available in Lozenge Form

• morphine sulfate

• lorazepam

• haloperidol

• clotrimazole

• nystatin

• diphenhydramine

• metoclopramide

• dexamethasone

• benztropine mesylate

Liquid Dosage Forms

The liquid dosage forms for oral use include syrup, elixir, and extract.

• Syrup is a sweetened liquid that contains the drug, sugar, and fl avoring.

• Elixir is similar to a syrup but contains a relatively high percentage of

alcohol.

• Extract is the oil or active portion of a plant or herb that is usually

removed, or extracted, with alcohol (e.g., an oil of peppermint or

wintergreen).

Liquid dosage forms

include syrup, elixir,

extract, tincture, solution,

and suspension.

Solutions and Suspensions

If the drug dissolves completely into the liquid (e.g., syrup, elixir), it is called

a solution. Another oral dosage form is the drug suspension, which is composed

of water and drug particles that do not dissolve but remain suspended

in the water. Suspensions need to be handled carefully, as the drug particles

tend to sink to the bottom very quickly. Mixing and drawing the dose can be

tricky—the withdrawal of the drug dose must be done immediately after mixing,

before the drug particles have a chance to settle. If the suspension is not

properly mixed or the dose is not drawn immediately, the wrong dose of drug

may be dispensed. If the dose is taken from the top of the container, it may

contain too much water and not enough drug. If it is taken from the bottom,

the drug solution may be too concentrated because the drug particles tend

to sink. In addition to mixing the suspension thoroughly, how the dose is

withdrawn matters, as well. The dose must be drawn up quickly, as the drug

particles may settle while the dose is being drawn.

Tincture

Tincture is another liquid dosage form. In modern times, it is only used

topically. The tincture is an alcohol-based drug form, such as tincture of

merthiolate, and is normally dispensed in a dropper bottle. These drugs are

not to be taken internally.

Drugs in suspension

need to be handled

carefully, as drug

particles may settle to

the bottom of the container

while the dose

is being withdrawn!

Semisolid Dosage Forms

The semisolid dosage forms include creams, lotions, ointments, and

suppositories.

• Creams and lotions are nothing more than emulsions (oil droplets suspended

in water), where the drug is usually dissolved in the oil. Creams

are thicker, as they contain less water than lotions.

• Ointments may vary from a thick emulsion to a drug suspended in a

waxy base, like petrolatum (which is like petroleum jelly, only much

stiffer and thicker). These preparations are usually used topically (on the

skin or mucous membranes, such as those in the mouth, inside the nose,

or rectum) and are normally dispensed in a tube or jar.

• Suppositories are made of wax and oils, and contain the drug that is meant

to be released slowly, and in a particular place. They are normally inserted

into body cavities, such as the rectum or vagina, where they adhere to the

cavity wall and release medication to the immediate area. Rectal suppositories

are also used to medicate patients who cannot take medication orally

(e.g., a vomiting patient), as the medication, if properly prepared, can be

absorbed through the rectal wall into the bloodstream. Suppositories are

normally large, and, being primarily made of soft wax, will melt at body

temperature. They should be stored in a cool room or refrigerated

(depending on the drug), and handling should be kept to a minimum

Storing Emulsions

Care must be taken when storing emulsions. Freezing the emulsion or exposing

it to excessive heat (near a heat source, for example, or storage in a warm room

for a long time) will cause the cream to separate into oil and water. Emulsions

should not be stored in the refrigerator and especially should never be frozen,

as the rapid change in temperature will cause the product to separate faster.

Emulsions should

never be frozen or

exposed to heat!

Administering the Drug—The Route of Administration

The route of administration defi nes how the drug gets into the body. Drugs

to be administered by different routes are prepared in different ways. The

most common route of administration is by mouth (oral, or po). These drugs

are given as a tablet or oral solution. Sublingual tablets (SL) are made to

dissolve under the tongue; the underside of the tongue and the fl oor of the

mouth contain large amounts of blood vessels near the surface, which allow

the drug to be absorbed into the system very quickly. These tablets are very

soft and dissolve easily. Sublingual preparations are also marketed in a spray

formulation, which are sprayed under the tongue.

Routes of administration include the following:

• Intranasal: a drug in drop or spray form is used

• Transdermal: a drug “patch” is used, which slowly releases drug into

the skin, where it is picked up by surface blood vessels and absorbed

into the body

• Inhalants: drugs may be used in powder or liquid form, in combination

with an inhalant apparatus, to be taken directly into the lungs

(e.g., drugs used for asthma)

• Administration through body cavities: drugs may be used in cream or

suppository form. They are inserted into body cavities, such as the

vagina or rectum, and used for local administration (e.g., for a yeast

infection or a case of hemorrhoids, respectively). Rectal administration

is also very useful for administration of drugs to a patient who cannot

take medications orally, as the drug is absorbed through vessels in the

rectal wall.

Drugs may also be administered through the lining of the cheek. This is

termed buccal (bYOUcahl) administration. The dosage form, in a lozenge or

buccal tablet, is inserted between the cheek and the gum.

Medicating the Eye and Ear

Drugs for the eye (ophthalmics) or ear (otics) are administered by drop (gtt).

The dropper or dropper container is calibrated to give a drop of the particular

size needed to give an accurate dose of drug.

Ophthalmic ointments may also be used (e.g., antibiotic ointments) and

are applied to the inside of the eyelid (usually at the bottom of the eye). The

tip of the ointment tube should never touch the eye.

Figure 2-2: Sterile instillation of eye medication

Parenteral Drug Administration

Any drug that is not given through the digestive system is given parenterally

(para means “around” and enteral refers to the digestive system). In

normal medical terms, however, parenteral administration refers to drugs

administered by injection. The three most common types of injections

are the intravenous, intramuscular, and subcutaneous injections. Other

types of injections include the intra-arterial, intracardiac, intrathecal, and

intradermal injections.

Injectable Drugs

Injections vary according to type. Intravenous injections are prepared in

three ways:

• The bolus: a one-time single-dose injection

• The IV drip: a bag or bottle of liquid that allows drug to be infused

over a long period of time (Figure 2-3)

• The “piggyback” IV: a solution contained in a smaller IV bag that is

infused along with the primary intravenous drip, usually through the

same tubing (Figure 2-4)

Intravenous injections

are seen in three

forms—the IV bolus,

IV drip, and “piggyback”

IV.

Intramuscular Injections

Intramuscular injections are placed into skeletal muscle. This allows the drug

to enter the bloodstream more slowly. This type of injection must fi rst diffuse

through muscle tissue before entering the bloodstream, so it requires a largebore

needle in order to penetrate the muscle.

The advantage to this type of injection is that the slow release of drug

into the system minimizes shock to the system, allowing it to gradually acclimate

to the effects of the drug.

Subcutaneous and Intradermal Injections

Injections into or under the skin include subcutaneous and intradermal injections.

Subcutaneous injections are placed under the skin, which allows for a slow

Figure 2-3: The IV Drip

When preparing an

intramuscular injection,

a large-bore needle

should be attached,

as a small needle will

not easily penetrate

muscle tissue.

absorption of drug into the bloodstream. Intradermal (ID) injections, which

are less common, are placed within the skin layers. Both of these types of injections

must be dispensed with a very fi ne needle (25–31 gauge) on the syringe.

Specialized Injections

Intra-arterial Injections. Occasionally, drugs need to be administered directly

into an artery, in order to have the best eff ect. Th ese are called intra-arterial injections.

Arteries are very muscular and the blood within them is under very high

pressure, so these injections require a somewhat larger bore needle.

Intrathecal and Intracardiac Injections. Intrathecal and intracardiac injections

are specialized injection forms. Intrathecal injections are placed into the

space between the spinal cord and spinal meninges (e.g., an epidural anesthetic

during childbirth), and intracardiac injections are placed directly into

the heart. These types of injections allow fast action of a drug by placing the

drug at the site of the organ itself.

Primary IV

Secondary IV

Figure 2-4: The Piggyback IV

Intramuscular and

subcutaneous injections

provide for a

slow rate of delivery of

drug to the system.

Interpreting the Prescription Order

Before fi lling the prescription order, you must fi rst check the prescription

form to make sure that the order is genuine, legal, and complete. Certain

information must be on the prescription form when it is received, and other

information may be fi lled in by the technician, unless the prescription is for a

controlled substance. In this case, no information is to be added, deleted, or

corrected on the prescription form.

Table 2-1 lists abbreviations commonly used on the prescription form

by the prescriber. These abbreviations must be interpreted accurately to

ensure that the correct medication is dispensed and that accurate instructions

are provided to the patient for the use of the medication. Additional

abbreviations may be found in Appendix A. You may be asked about any

of these, even abbreviations seldom used, on the exam, so it is wise to be

familiar with them.

Figure 2-5 represents the prescription form that would be received at the

pharmacy window. Information required to correctly fi ll this order is found

in the body of the prescription. Review the information required to appear

on the prescription:

• The drug name: This can be generic (the actual name of the drug) or a

brand (proprietary) name. This prescription specifi es the exact drug to

select for dispensing. This prescription was written for a brand name,

Lasix, although the prescriber did sign on the “May Substitute” line, so

generic substitution is permissible.

• The strength and dosage form of the drug: Drugs come in different

strengths and forms for different needs. The strength and form must

be specifi ed, unless the drug comes in only one form or strength. For

example, some combination drugs such as trimethoprim with sulfamethoxazole

combination or acetaminophen with codeine (Tylenol

#3, etc.) are dispensed in a specifi c dosage and proportion. Mannitol is

dispensed only in a solution for injection. The proportions and forms

of these drugs do not need to be specifi ed on the prescription form. In

contrast, Lasix tablets come in 20 mg, 40 mg, and 80 mg strengths, as

well as in oral solution and solution for injection. The dosage strength

Drugs are dispensed in

diff erent dosage forms

for diff erent needs.

John Smith M.D.

201 Tablet Lane

Anywhere USA

DEA# AS274064

Name

Address

Dispense as Written

Refill 0 1 2 3 4 5

SIG:

T

Date

May Substitute

Sally Swollen

John Smith M.D.

2/1/XX

Lasix 40 mg tabs #60

BID PRN edema

Figure 2-5: Sample Completed Prescription Form

and form did need to be specifi ed in the sample prescription shown in

Figure 2-5.

• The amount of drug prescribed: A prescription for tablets, such as that

in Figure 2-1, must specify the number of tablets to be dispensed. For

other dosage forms, however, this may not be the case. For example, a

prescription for a liquid dosage form may be specifi ed in more than one

way. Either the volume may be specifi ed, or the drug dose may be specifi

ed in mg, g, and so on.

EXAMPLE

The prescription order is for 500 mL of 10% calcium gluconate solution.

Since the volume was given, the specifi ed amount of solution (500 mL)

would be dispensed.

EXAMPLE

The prescription order is for 200 mg of Minocin IV. Minocin comes in a

sterile solution of 20 mg/mL. In this case, the volume of solution to be

dispensed for a 200 mg dose would have to be calculated (e.g., 200 mg

divided by 20 mg  10 mL).

• Instructions for the patient (the SIG): This is where knowledge of the

abbreviations in Table 2-1 comes in. Since the instructions must be

written out for the patient, the technician must be able to accurately

read the SIG. The prescription in Figure 2-5 states that one tablet

(designated by a horizontal bar with one vertical bar and one dot) is to

be taken twice a day (bid, or bis in deum), as needed (prn) for edema.

The amount of medication to be taken, and limitations on when or how

often it is to be taken, must be included on the prescription form.

The spacing of the doses, or dosage interval, is extremely important, as

the space between doses is based on the half-life (T1/2) of the drug. The T1/2

is a measure of how rapidly a drug is cleared from the body, and gives an

estimate of how quickly the effects of the drug will be terminated. (There

are many ways in which the actions of a drug may be terminated, but the

half-life is generally considered to be the main index of the length of a

drug’s effects.)

The half-life can be used to predict the dosage interval for a drug. To keep

the serum levels of a drug relatively constant, the drug should be replaced as

it is cleared from the body. Thus, dosage intervals are very important, and

the instructions for taking the drug must be communicated effectively to the

patient. It is also important to communicate to the patient the proper use of

the drug (e.g., proper insertion of a suppository, instillation of an ophthalmic

preparation, etc.).

The half-life of a drug

is the amount of time

taken for half of the

serum concentration

of drug to be eliminated

from the body.

It is used to establish

accurate dosage

intervals.

A drug dose may be

specifi ed by volume or

by equivalent weight

of drug.

EXAMPLE

The time it takes a drug to be eliminated from the body is around 5–7

half-lifes. If a drug has a 6-hour half-life, then it would take 30–42 hours

to be eliminated. (6 hrs  5  30; 6 hrs  7  42.)

• Signature of the prescriber and authorization to substitute: The signature

must be handwritten in ink. The authorization to dispense a generic

drug may be indicated in a box on the prescription form, in which the

letters “DAW” (“dispense as written”) are written (indicating that the

exact proprietary label must be dispensed) or absent (indicating that a

substitution is permissible). Depending on the state, the prescription

form may contain this box or may have a duplicate set of signature lines

bearing a designation such as “may substitute” or “no substitution permissible.”

If the prescriber designates “no substitution permissible,” the

drug must be dispensed exactly as written, in the correct form, strength,

and under the specifi ed proprietary label.

Information is normally entered on the prescription form by the technician

and then transferred to the patient profi le. Information to be gathered

includes the following:

• The patient’s address and telephone number: This information identifi es

the patient (there may be more than one patient with the same name).

It also provides a means of contact with the patient, in case of a problem

with a prescription or drug recall.

• The age or date of birth of the patient: This information is very important,

as it serves to identify the patient (e.g., to distinguish between a

father and son with the same name) and assures that the drug dosage

prescribed is appropriate for the age of the patient (drug dosage may be

reduced in a child or elderly person, for example, as organ functions are

less effi cient).

• Drug allergies: Many drugs are very similar in chemical structure and action.

Thus, if a patient is allergic to one drug (e.g., penicillin), he or she

may well be allergic to similar drugs, such as amoxicillin or even cephalexin.

A history of drug allergies is critical to the care of the patient, as it

may help prevent an uncomfortable or even fatal allergic reaction.

• Concurrent medications: These are medications already being taken by

the patient. A history of concurrent medications should include not

only other prescription medications but also those purchased over the

counter (e.g., cold remedies), and herbal remedies as well. (The fi rst

drugs were little more than pulverized plants, or plant extracts, after

all. We have done little more than refi ne them, in many cases.) Herbal

preparations can have very potent drug actions and interactions and

must be recorded in the patient profi le.

The “may substitute”

option gives the

patient and pharmacy

the option to choose a

less expensive generic

brand or another proprietary

label, as long

as the drug, strength,

and form remain the

same.

Many drugs interact

with each other to produce

adverse eff ects.

A particular drug may

also greatly increase

the therapeutic effects

of another drug,

which would require

an adjustment to the

patient’s dosage.

Dispensing the Correct Medication

Once the drug, dosage form, and strength have been established, the correct

medication is selected. This medication should be exactly what appears on the

prescription form.

Verifying the Medication—Use of the Manufacturer’s Label

Many drug names look alike and sound alike, so the manufacturer labels must

be compared carefully to the prescription order.

EXAMPLE

Extra letters may be present in the drug name on the label (e.g., Adalat

CC instead of Adalat). This may mean the drug is a different formulation

of the brand-name drug (in this case an extended-release form) or

may be a different drug altogether (e.g., quinine and quinidine). Some

of those abbreviations can be found in Table 2-3. If the name of the

drug does not match exactly, the drug should not be dispensed.

Verifying the Proper Dosage Strength

The choice of dosage strength is less critical than other information. If the

dosage strength does not match, it may be possible to convert dosages

(see Chapters 4 and 14). If the dosage form is incorrect, however, the drug

cannot be dispensed by the technician without consulting the pharmacist.

Table 2-3 Extended-release Formulations

LA long acting

SA sustained acting

SR sustained release

TR timed release

ER extended release

EXAMPLE

The drug order is for 250 mg amoxicillin tablets. There are no tablets

in stock, but the pharmacy does have amoxicillin suspension in stock

for oral administration. Both dosage forms are for oral administration,

so the suspension could be substituted, with proper calculations and

patient instruction (this would require the approval of the pharmacist).

EXAMPLE

The drug order is for Compazine suppositories. You have Compazine

solution for oral administration in stock, but no suppositories. The

order cannot be fi lled, as the dosage forms do not match (suppositories

are normally prescribed for patients who cannot take medications

orally).

Automated Unit Dose Delivery Systems

There are several automated dispensing systems presently marketed for institutional

use. One popular and innovative automated unit dose delivery

system coming into widespread use in institutional pharmacy is the Pyxis Rx

System. The Pyxis system is essentially a computerized cabinet that is located

on a hospital fl oor (unit). The cabinet is stocked with drugs, which are appropriate

to the particular hospital unit where it is located. Like the med

cart, drugs are fi led in locked drawers within the cabinet, and the units are

maintained and stocked by pharmacy personnel. The computer within the

Pyxis unit is on a local area network, which interfaces with the main hospital

computer. Thus, the unit actually charts patient medications as they are withdrawn

from the cart by hospital personnel.

Processing of Medication Orders Using the Pyxis System

The Pyxis system streamlines the dispensing of medication. Medication orders

are received as usual from physicians in the pharmacy. The pharmacy technician

then enters the orders into the main hospital computer system. The orders are

then checked by the pharmacist to ensure that the medications and doses are

appropriate for the age, weight, and diagnosis of the patient, and that therapeutic

duplications and drug-drug interactions are not present. The order is

then sent to the Pyxis system. Once the order has been verifi ed and is present

in the system, the fl oor nurse can enter appropriate information into the system

when it is time for a patient’s medication. The system then allows the withdrawal

of the proper unit doses of medication for administration to the patient.

Identifi cation of the nurse, by thumbprint or code, must be received by the

unit for the medication drawers to unlock and the medication to be withdrawn.

Advantages to the Use of Automated Unit Dosing Systems

The advantages to this system are many: Medication errors are reduced, as

the medication dispensed comes directly from the original medication order

(i.e., not faxed, transcribed, or photocopied); drug-drug interactions are

reduced; and patients receive their medications in a more timely manner, allowing more effective dosing. In addition, input from the pharmacist is almost

instantaneous. Blood analysis of drug levels can also be included in the

computerized information, allowing dosages to be adjusted almost instantaneously.

This provides better control over patient medication. Also, as patients

are transferred from room to room and fl oor to fl oor, their information

remains centralized with less chance of record loss. Documentation of drug

dispensing and administration is generated automatically with the system,

and can be printed out at any time, should a hard copy be needed.

Comparison of Drug Dispensing in Retail and Institutional Settings

Dispensing a prescription in an institutional setting is similar to the retail

setting, with a few exceptions. Several drugs are usually prescribed at once

(see Chapter 1) using the hospital order; these doses may be sent up to the

patient individually (e.g., a medication needed quickly, for an emergency

[STAT], or a medication prescribed for pain, emesis, etc., which is not part

of the usual routine of drugs), or placed into a unit dose cart. Unit dose

carts contain the daily medications of the patients on a particular hospital

fl oor. They are prepared daily by technicians and then checked by pharmacists.

These computerized carts contain the individual medications of

patients on the fl oor, normally enough to last for one day. The carts are

fi lled daily, from the physician’s orders for the various patients on the fl oor,

making it easier for nurses to properly administer medications to patients.

Narcotics prescribed “as needed” may not be dispensed in a unit dose cart.