Alkanes, Cycloalkanes, and Conformations — Study Notes

Organic molecules: hydrocarbons, alkanes, and basic nomenclature

  • Organic compound definition: a compound that contains carbon, with carbon as the central atom; if the compound also has hydrogen attached to carbon, it’s an organic compound.

    • Hydrocarbon: an organic compound that contains only carbon and hydrogen (no oxygen, nitrogen, etc.).

    • Distinction: carbohydrates (e.g., sugar) are different from hydrocarbons (e.g., hydrocarbons are generic name for carbon–hydrogen compounds without other heteroatoms).

  • Alkane basics (a subfamily of hydrocarbons):

    • Alkanes are hydrocarbons with only single bonds between carbon atoms; all carbons are sp^3 hybridized.

    • sp^3 hybridization meaning: carbon forms four single bonds (to four substituents, which can be hydrogen or carbon). No double or triple bonds.

    • Consequence: each carbon in an alkane forms only single bonds; no pi bonds in the backbone.

  • Simple alkanes: naming and basic structures

    • Methane (CH4): carbon at center with four hydrogens (CH4).

    • Ethane (C2H6): backbone of two carbons, each bonded to three hydrogens; all hydrogens and carbons are saturated; formula: C<em>2H</em>6C<em>2H</em>6.

    • Propane (C3H8): carbon backbone of three; end carbons each have three hydrogens, middle carbon has two hydrogens; formula: C<em>3H</em>8C<em>3H</em>8.

    • Butane (C4H10): straight-chain (acyclic) or branched forms exist; condensed forms shown, e.g., CH3-CH2-CH2-CH3 or CH3-CH(CH3)-CH_3 (isobutane).

    • General condensed Lewis structures: show carbon centers with attached hydrogens; Lewis structure emphasizes bonding electrons; for hydrocarbons, all electrons are involved in bonding (no lone pairs on C or H).

  • General formula for acyclic (non-cyclic) alkanes

    • For an alkane with n carbons: C<em>nH</em>2n+2C<em>nH</em>{2n+2}

    • This arises because each carbon needs four bonds; in a straight chain, there are two terminal carbons contributing 3 hydrogens each and internal carbons contributing 2 hydrogens; overall lead to 2n+2 hydrogens.

    • Example checks: n=1 (CH4) gives H4; n=2 (C2H6) gives H6; n=3 (C3H8) gives H8; n=4 (C4H{10}) gives H_{10}.

  • Constitutional isomers of alkanes (same formula, different connectivity)

    • Pentane (C5H{12}) has three constitutional isomers:

    • n-pentane (a straight chain),

    • isopentane (2-methylbutane),

    • neopentane (2,2-dimethylpropane).

    • All three share the same molecular formula but differ in carbon connectivity; they are constitutional (structural) isomers.

    • For C5H{12}, these three are explicitly illustrated in class notes:

    • n-pentane: CH3-CH2-CH2-CH2-CH_3

    • isopentane (2-methylbutane): CH3-CH(CH3)-CH2-CH3

    • neopentane (2,2-dimethylpropane): a central quaternary carbon bound to four CH_3 groups

    • General idea: different ways to arrange the same number of carbons and hydrogens yield constitutional isomers; these are non-identical in bonding pattern but identical in formula.

  • Condensed Lewis structures versus full drawings

    • Condensed Lewis form vs full Lewis structure: condensed form lists the atoms and their immediate attachments (e.g., CH3-CH2-CH_3), while full Lewis structures show all bonds and electron pairs.

    • For butane (C4H{10}) you can present as:

    • Linear: CH3-CH2-CH2-CH3

    • Branched (isobutane): CH3-CH(CH3)-CH_3

    • The condensed form helps visualize connectivity; full Lewis shows bonding electrons explicitly; both describe the same molecule.

  • Short-hand (skeletal) representations and cautions

    • In shorthand, carbons are at endpoints and intersections; hydrogens on these carbons are generally not drawn, unless the molecule is very small.

    • For example, butane often written as CH3-CH2-CH2-CH3 or as a zigzag with implicit hydrogens; shorthand helps readability for larger molecules.

  • General formula for monocyclic alkanes (cycloalkanes)

    • Monocyclic alkanes are alkanes with one ring; formula differs from acyclic by ring closure.

    • General formula for monocyclic alkanes: C<em>nH</em>2nC<em>nH</em>{2n}

    • Smallest monocycle: cyclopropane (C3H6).

    • Examples: cyclobutane (C4H8), cyclopentane (C5H{10}), cyclohexane (C6H{12}).

    • In cycloalkanes, every carbon is sp^3 hybridized and the ring closes by removing two hydrogens to form a C–C bond that completes the ring.

  • Cycloalkane naming and substituents

    • Nomenclature basics: prefix cyclo- is added to the base name of the ring (e.g., cyclopentane).

    • If there is one substituent on the ring, you usually do not need to specify the number 1 (e.g., methylcyclopentane).

    • If there are multiple substituents, or substituents on different carbons, numbers are assigned to give the lowest set of locants, and substituents are named in alphabetical order (ignoring prefixes like di-, tri-, etc., and ignoring cyclo in alphabetizing but including iso- when applicable).

    • For cycloalkanes with multiple substituents, the substituents can be placed on different ring carbons, and the substituent numbers are chosen to minimize the sum of locants; for example, 1-ethyl-3-methylcyclopentane vs other possible placements.

  • Substituent naming: alkyl groups derived from alkanes

    • Replace one H on an alkane with a substituent (an alkyl group): alkyl groups attach to the parent chain.

    • Common alkyl groups (with their formulas when attached):

    • Methyl: —CH3 (from methane, CH4)

    • Ethyl: —CH2CH3 (from ethane, C2H6)

    • Propyl: —CH2CH2CH3 (from propane, C3H_8)

    • Isopropyl: —CH(CH3)2 (propyl isomer, same formula as n-propyl but different connectivity)

    • Butyl: —C4H9 (from butane, C4H{10})

      • Secondary butyl (sec-butyl): attachment from a secondary carbon

      • Isobutyl: (CH3)2CHCH2–

      • Tert-butyl (t-butyl): attachment from a tertiary carbon

    • Important notation and prefixes:

    • The IUPAC substituent prefixes include isopropyl, isobutyl, sec-butyl, tert-butyl, etc.

    • When alphabetizing substituents, drop prefixes such as di- and tri-, and drop secondary/tertiary prefixes for alphabetization; iso- remains part of the name (e.g., isopropyl, isobutyl).

    • For multi-substituent compounds, use prefixes like di-, tri- in the name to indicate multiple identical substituents on different carbons (e.g., 2,2-dimethyl).

  • Examples of substituent naming on alkanes

    • Propane derivatives: two different propyl isomers are formed when attaching a substituent to a propane molecule depending on which hydrogen is removed; substituents include propyl and isopropyl.

    • Butane derivatives: possible substituents include butyl (on terminal carbon) and sec-butyl (on either terminal or internal carbon), with isobutyl and tert-butyl providing other attachment patterns.

    • The IUPAC approach: identify the longest carbon chain (the parent), then name substituents on that chain with lowest locants, then order substituents alphabetically (ignoring prefixes like di/tri and ignoring cyclo when discussing cyclic systems, but including iso-prefixes when applicable).

  • Steps to name an alkane (acyclic)

    • Step 1: Find the longest continuous carbon chain. This becomes the parent chain (backbone).

    • Step 2: If there are multiple chains with the same maximum length, choose the one with the greater number of substituents (to keep substituents light and to minimize locants).

    • Step 3: Number the carbons in the parent chain from the end that gives the first substituent the lowest possible locant; if there is a tie, choose the direction that gives the next substituent the lowest locant, and so on.

    • Step 4: List substituents in alphabetical order, ignoring prefix di-, tri-, sec-, tert-, etc. Keep iso- prefixes in the alphabetization.

    • Step 5: If identical substituents occur on the same carbon, assign separate locants (e.g., 2,2-dimethyl).

    • Step 6: If a substituent is multiple atoms long, write its name before the parent chain name (e.g., 4-ethyl-2-methylhexane).

    • Step 7: Use hyphens to separate locants from substituent names and from the parent chain name; use a comma to separate multiple locants (e.g., 2,3-dimethylpentane).

  • Example naming walkthroughs

    • Example 1: Butane (C4H{10})

    • Longest chain: 4 carbons → butane (or butane-1? no, usually just butane; if branched, e.g., methylpropane is isobutane, etc.).

    • If branched to give two methyl groups on the second and third carbons: 2,2-dimethylpropane (neopentane) is a constitutional isomer of C5H{12}.

    • Example 2: Pentane derivatives

    • n-pentane: no substituents, just a five-carbon chain.

    • 2-methylbutane (isopentane): methyl substituent on carbon 2.

    • 2,2-dimethylpropane (neopentane): two methyl groups on the central carbon of the propane backbone.

  • Cycloalkanes: naming and numbering rules

    • Cycloalkanes are carbons arranged in a ring; the base formula is CnH{2n}.

    • For monocyclic cycloalkanes with one substituent: name as substituent-cycloalkane (e.g., methylcyclopentane); no need to prefix 1-.

    • If there are multiple substituents:

    • Number the ring to give substituents the lowest set of locants.

    • Use cyclo- in the base name; list substituents in alphabetical order, ignoring cyclo- and any numerical prefixes (e.g., cyclohexane with substituents ethyl and methyl would be 1-ethyl-3-methylcyclohexane, with ethyl listed before methyl).

    • When there are multiple identical substituents on the ring, use di-, tri-, etc., to indicate multiplicity and specify their positions (e.g., 1,3-dimethylcyclohexane).

    • In nomenclature examples given: cycloheptane, cyclopropane, cyclobutane, cyclohexane, cyclopentane, etc.

  • Conformational analysis of alkanes: rotation about C–C single bonds

    • Alkanes are free to rotate around C–C single bonds due to the sigma (σ) bond overlap of sp^3–sp^3 orbitals (no pi-bond lock).

    • Consequences: different spatial arrangements (conformations) of the same molecule can interconvert without breaking bonds.

    • Conformations are different spatial arrangements around a C–C bond; rotation changes how substituents are oriented in space, but not connectivity.

  • Ethane conformations: eclipse vs staggered

    • Two extreme conformations for ethane: eclipsed (or eclipsed ethane) and staggered.

    • Eclipse: hydrogens on adjacent carbons align with each other (front and back hydrogens are directly in line); there is more steric repulsion.

    • Staggered: hydrogens on adjacent carbons are offset from each other, reducing steric repulsion and lowering energy.

    • The energy difference between eclipsed and staggered conformations is about riangleE<br>oughly3extkcal/molriangle E <br>oughly 3 ext{ kcal/mol}, with staggered being more stable.

  • Dihedral angle and conformations

    • The dihedral angle (θ) is the angle between a substituent on the front carbon and the corresponding substituent on the back carbon as you rotate around the C–C bond.

    • Key angular positions in the staggered/eclipsed sequence occur at 0°, 60°, 120°, 180°, 240°, 300° (or 0°, 60°, 120°, 180°, 240°, 300° depending on the reference).

    • In Newman projections, the front carbon is drawn as the center, with the back carbon rotated to show relative positions of substituents around the C–C bond.

    • In sawhorse representations, you show a three-dimensional sense with wedges and dashes to indicate coming out of or going into the plane.

  • Visual representations: sawhorse and Newman projections

    • Sawhorse representation: shows bonds in 3D with planes and dashed/wedged bonds to indicate substituents coming out of or going behind the plane; useful for visualizing actual 3D orientation.

    • Newman projection: view down the C–C bond; front carbon at the center; back carbon at the circumference; substituents placed around; allows easy read of dihedral angles (0°, 60°, 120°, 180°, etc.).

    • Dihedral angles and conformational energies can be tracked by rotating one substituent around the C–C bond while keeping the other fixed.

  • Relative stability and energy profile of conformations

    • The eclipsed conformation is less stable (higher energy) due to steric repulsion between adjacent hydrogens (or substituents).

    • The staggered conformation is more stable (lower energy) because substituents are anti-periplanar and minimize repulsive interactions.

    • When rotating from eclipsed to staggered, energy drops by about riangleE<br>oughly3extkcal/mol.riangle E <br>oughly 3 ext{ kcal/mol}.

    • The energy profile for rotation about a C–C single bond typically shows repeating cycles of high-energy eclipsed peaks and low-energy staggered troughs every 60°.

  • Going from simple to more complex conformations (future topics)

    • In larger alkanes, the bulkiness of substituents (e.g., tert-butyl, isopropyl, etc.) affects the energy landscape and preferred conformations.

    • In later chapters, stereochemistry and more advanced conformational analyses (including substituted alkanes) will be discussed.

    • If given a molecular weight, you can determine the number of carbons using the general formula and the atomic weights: C = 12, H = 1; for an alkane: $$CnH{2n+2} \